SCHEMBL6893946

SCHEMBL6893946

CC(C)(C)c1c(O)ccc(C#N)c1C(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
AR P10275 14/20 0.40
PGR P06401 4/20 0.36
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36
ALDH1A1 P00352 2/20 0.34
ALOX15 P16050 2/20 0.34
HSD17B10 Q99714 2/20 0.34
HPGD P15428 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
UPP1 Q16831 1/20 0.34
NR1I2 O75469 1/20 0.33
LMNA P02545 1/20 0.33
CYP2C9 P11712 1/20 0.33
MIF P14174 1/20 0.33
TYR P14679 1/20 0.33
HTT P42858 1/20 0.33
NFE2L2 Q16236 1/20 0.33
ESR2 Q92731 1/20 0.33
SNCA P37840 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17030752 0.82 AR (0.39) ARPGRALDH1A1TDP1HTT
SCHEMBL8768208 0.79 ALDH1A1 (0.34) ALDH1A1ALOX15HSD17B10HPGDTDP1
SCHEMBL27963029 0.79 ALDH1A1 (0.48) ARALDH1A1ALOX15HSD17B10HPGD
SCHEMBL30027143 0.79 ALDH1A1 (0.48) ARALDH1A1ALOX15HSD17B10HPGD
SCHEMBL70068 0.79 ALDH1A1 (0.48) ARALDH1A1ALOX15HSD17B10HPGD
SCHEMBL26259842 0.76 AR (0.40) ARPGRALDH1A1
SCHEMBL20143843 0.73 TSHR (0.46) ARALDH1A1CYP2C9HTT
Hydroquinone SCHEMBL28076397 0.72 LMNA (0.55) ARALDH1A1ALOX15HSD17B10HPGD
SCHEMBL5694506 0.72 ALDH1A1 (0.42) ARALDH1A1ALOX15HSD17B10HPGD
Water SCHEMBL28289219 0.71 ESR1 (0.41) ARALDH1A1ALOX15HSD17B10HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1126833-A4 OXADIAZOLE, THIADIAZOLE AND TRIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF TREGA BIOSCIENCES INC (US) 2004-09-08 EP disclosed
EP-1150565-A1 THIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF LION bioscience AG (DE) 2001-11-07 EP disclosed
EP-1126833-A2 OXADIAZOLE, THIADIAZOLE AND TRIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF TREGA BIOSCIENCES, INC. (US) 2001-08-29 EP disclosed
WO-2000045635-A1 THIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF LION BIOSCIENCE AG (DE) 2000-08-10 WO disclosed
WO-2000025768-A1 OXADIAZOLE, THIADIAZOLE AND TRIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF TREGA BIOSCIENCES, INC. (US) 2000-05-11 WO disclosed