SCHEMBL6895096

SCHEMBL6895096

O=C(OCBr)Oc1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.44
TDP1 Q9NUW8 2/20 0.44
KDM4E B2RXH2 1/20 0.44
ATM Q13315 2/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
ALOX15 P16050 2/20 0.43
HSD17B10 Q99714 2/20 0.42
HPGD P15428 1/20 0.42
ALDH1A1 P00352 1/20 0.42
CYP19A1 P11511 1/20 0.42
MEN1 O00255 1/20 0.41
HTT P42858 1/20 0.41
GFER P55789 1/20 0.41
KMT2A Q03164 1/20 0.41
PTPN1 P18031 1/20 0.40
GSK3B P49841 1/20 0.40
NSD2 O96028 1/20 0.40
USP2 O75604 1/20 0.40
MTNR1A P48039 1/20 0.39
MTNR1B P49286 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10835857 0.86 MAPT (0.41) MAPTTDP1KDM4EATML3MBTL1
SCHEMBL10025073 0.84 MAPT (0.46) MAPTTDP1KDM4EATML3MBTL1
SCHEMBL8646552 0.84 THRB (0.47) MAPTTDP1KDM4EATML3MBTL1
SCHEMBL28211567 0.84 MAPT (0.40) MAPTTDP1KDM4EATML3MBTL1
SCHEMBL10025075 0.83 MAPT (0.44) MAPTTDP1KDM4EATML3MBTL1
SCHEMBL322125 0.83 MAPT (0.44) MAPTTDP1KDM4EATML3MBTL1
SCHEMBL9353455 0.81 TDP1 (0.54) MAPTTDP1KDM4EATML3MBTL1
SCHEMBL18073 0.81 TDP1 (0.54) MAPTTDP1KDM4EATML3MBTL1
SCHEMBL9353461 0.81 TDP1 (0.54) MAPTTDP1KDM4EATML3MBTL1
SCHEMBL27352197 0.81 TDP1 (0.54) MAPTTDP1KDM4EATML3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1392312-A1 TRIAZOLO 4,5-d] PYRIMIDINE DERIVATIVES AND THEIR USE AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2004-03-03 EP disclosed
WO-2002055083-A1 TRIAZOLO[4,5-d] PYRIMIDINE DERIVATIVES AND THEIR USE AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2002-07-18 WO disclosed