SCHEMBL6895340

SCHEMBL6895340

COc1ccc(CN=C=O)cc1.COc1ccc(N=C=O)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MIF P14174 1/20 0.56
CYP3A4 P08684 2/20 0.50
TSHR P16473 1/20 0.50
MPI P34949 1/20 0.41
APLNR P35414 1/20 0.39
IDO1 P14902 2/20 0.39
CYP1A2 P05177 1/20 0.39
MAPT P10636 3/20 0.38
TRPA1 O75762 1/20 0.38
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
ALOX15 P16050 1/20 0.38
CMA1 P23946 1/20 0.38
PYCR1 P32322 1/20 0.37
AGXT P21549 1/20 0.37
LTA4H P09960 1/20 0.37
TAAR1 Q96RJ0 1/20 0.37
HTT P42858 2/20 0.37
LDHA P00338 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5372 0.90 MIF (0.67) MIFCYP3A4TSHRMPIAPLNR
SCHEMBL302097 0.86 CYP3A4 (0.65) MIFCYP3A4TSHRCYP1A2TRPA1
SCHEMBL161063 0.84 CYP3A4 (0.50) CYP3A4TSHRMAPTTRPA1ALDH1A1
Phenylacetic Acid SCHEMBL7876128 0.83 KDM4E (0.43) MIFMAPTKDM4EALDH1A1SMN1; SMN2
SCHEMBL9716383 0.81 CYP3A4 (0.59) MIFCYP3A4TSHRCYP1A2TRPA1
Methylene Chloride SCHEMBL28742344 0.81 CYP3A4 (0.48) MIFCYP3A4TSHRMAPTTRPA1
SCHEMBL27899734 0.81 CYP3A4 (0.59) MIFCYP3A4TSHRCYP1A2TRPA1
SCHEMBL29087457 0.81 CYP3A4 (0.59) MIFCYP3A4TSHRCYP1A2TRPA1
SCHEMBL13246064 0.79 ESR2 (0.47) CYP3A4TSHRMAPTALDH1A1SMN1; SMN2
SCHEMBL28101787 0.79 LTA4H (0.48) CYP3A4TSHRCYP1A2MAPTTRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1126833-A4 OXADIAZOLE, THIADIAZOLE AND TRIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF TREGA BIOSCIENCES INC (US) 2004-09-08 EP disclosed
EP-1126833-A2 OXADIAZOLE, THIADIAZOLE AND TRIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF TREGA BIOSCIENCES, INC. (US) 2001-08-29 EP disclosed
WO-2000025768-A1 OXADIAZOLE, THIADIAZOLE AND TRIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF TREGA BIOSCIENCES, INC. (US) 2000-05-11 WO disclosed