SCHEMBL6896587

SCHEMBL6896587

COc1cc(OC)c(C(=O)CCc2ccc(N)cc2)c(OC)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFKB1 P19838 1/20 0.58
NFKB2 Q00653 1/20 0.58
RELA Q04206 1/20 0.58
CYP19A1 P11511 5/20 0.55
SLC5A1 P13866 1/20 0.54
SLC5A2 P31639 1/20 0.54
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
CYP2D6 P10635 2/20 0.49
LMNA P02545 1/20 0.49
HTR1A P08908 1/20 0.49
ADRA2A P08913 1/20 0.49
ADRA2C P18825 1/20 0.49
OPRK1 P41145 1/20 0.49
KCNH2 Q12809 1/20 0.49
EBP Q15125 1/20 0.49
SIGMAR1 Q99720 1/20 0.49
HRH3 Q9Y5N1 1/20 0.49
F2RL1 P55085 1/20 0.46
MAPT P10636 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26528807 0.89 NFKB1 (0.72) NFKB1NFKB2RELACYP19A1SLC5A1
SCHEMBL17502354 0.85 RAB9A (0.60) NFKB1NFKB2RELASLC5A1SLC5A2
SCHEMBL6398047 0.83 NFKB1 (0.60) NFKB1NFKB2RELACYP19A1SLC5A1
SCHEMBL6398347 0.81 NFKB1 (0.74) NFKB1NFKB2RELACYP19A1SLC5A1
SCHEMBL2282039 0.81 NFKB1 (0.83) NFKB1NFKB2RELACYP19A1SLC5A1
SCHEMBL9578083 0.80 NFKB1 (0.59) NFKB1NFKB2RELACYP19A1SLC5A1
SCHEMBL7193907 0.79 CYP2D6 (0.57) NFKB1NFKB2RELACYP19A1SLC5A1
SCHEMBL11297508 0.79 NFKB1 (0.70) NFKB1NFKB2RELACYP19A1SLC5A1
SCHEMBL2978651 0.79 NFKB1 (0.66) NFKB1NFKB2RELACYP19A1SLC5A1
SCHEMBL29684688 0.79 NFKB1 (0.66) NFKB1NFKB2RELACYP19A1SLC5A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0674530-B1 RADIOLABELED POLYHYDRIC PHENOL COMPOUNDS MALLINCKRODT INC (US) 2004-09-01 EP disclosed
US-5780008-A DIAGNOSTIC AGENT FOR INCREASED GLUCOSE METABOLISM AND/OR FOR TUMOR CELLS; RADIOLABELLED DERIVATIVES OF PHLORETIN, GENISTEIN, NARINGENIN AHD PHLORIZIN; RADIOLOGY MALLINCKRODT MEDICAL, INC. (US) 1998-07-14 US disclosed
US-5741476-A RADIOLABELLED WITH HALOGEN ISOTOPE; MEDICAL DIAGNOSIS, ANTITUMOR AGENTS MALLINCKRODT MEDICAL, INC. (US) 1998-04-21 US disclosed