SCHEMBL6898504

SCHEMBL6898504

CCN(CC)CCOc1ccccc1NC(=O)c1ccc(Cc2ccccc2)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.56
DRD2 P14416 1/20 0.55
DRD1 P21728 1/20 0.55
DRD3 P35462 1/20 0.55
MCHR1 Q99705 6/20 0.54
CYP1A2 P05177 1/20 0.54
LTA4H P09960 1/20 0.54
CYP2D6 P10635 1/20 0.54
CYP2C9 P11712 1/20 0.54
CYP2C19 P33261 1/20 0.54
HTT P42858 1/20 0.54
CACNA1H O95180 1/20 0.49
CACNA1B Q00975 1/20 0.49
ALDH1A1 P00352 2/20 0.49
KDM4E B2RXH2 1/20 0.49
LMNA P02545 1/20 0.49
POLB P06746 1/20 0.48
TSHR P16473 1/20 0.48
P4HTM Q9NXG6 1/20 0.47
NPC1 O15118 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6898486 0.92 GAA (0.58) GAADRD2DRD1DRD3MCHR1
SCHEMBL3500701 0.91 GAA (0.60) GAADRD2DRD1DRD3MCHR1
SCHEMBL6927664 0.88 MCHR1 (0.61) GAAMCHR1CACNA1HCACNA1BALDH1A1
SCHEMBL7056986 0.86 CACNA1H (0.63) GAAMCHR1CACNA1HCACNA1BALDH1A1
SCHEMBL6925417 0.86 GAA (0.58) GAAMCHR1CACNA1HCACNA1BALDH1A1
SCHEMBL6898482 0.85 MCHR1 (0.68) GAAMCHR1LTA4HCACNA1HCACNA1B
SCHEMBL6926348 0.85 GAA (0.57) GAAMCHR1CACNA1HCACNA1BALDH1A1
SCHEMBL6927791 0.84 GAA (0.59) GAAMCHR1CACNA1HCACNA1BALDH1A1
SCHEMBL6808491 0.82 MCHR1 (0.69) MCHR1CYP1A2LTA4HCYP2D6CYP2C9
SCHEMBL6928305 0.80 MCHR1 (0.52) GAAMCHR1CACNA1HCACNA1BALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1100485-A4 SUBSTITUTED ANILIDE COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORP (US) 2004-06-09 EP claimed
JP-2002521436-A 2002-07-16 JP claimed
EP-1100485-A1 SUBSTITUTED ANILIDE COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2001-05-23 EP claimed
WO-2000006146-A9 SUBSTITUTED ANILIDE COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORP (US) 2000-08-03 WO claimed
WO-2000006146-A1 SUBSTITUTED ANILIDE COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2000-02-10 WO claimed
EP-1100485-A4 SUBSTITUTED ANILIDE COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORP (US) 2004-06-09 EP disclosed
EP-1100485-A1 SUBSTITUTED ANILIDE COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2001-05-23 EP disclosed
WO-2000006146-A9 SUBSTITUTED ANILIDE COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORP (US) 2000-08-03 WO disclosed
WO-2000006146-A1 SUBSTITUTED ANILIDE COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2000-02-10 WO disclosed