SCHEMBL6900513

SCHEMBL6900513

Bc1ccc(OCCN)c(C(F)(F)F)c1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.40
S1PR1 P21453 11/20 0.38
HTR2A P28223 1/20 0.37
HTR2C P28335 1/20 0.37
S1PR4 O95977 1/20 0.37
THRA P10827 1/20 0.34
THRB P10828 1/20 0.34
HTR1B P28222 1/20 0.34
ESR1 P03372 1/20 0.34
RXRA P19793 1/20 0.34
RXRB P28702 1/20 0.34
RXRG P48443 1/20 0.34
CTSS P25774 2/20 0.34
CTSK P43235 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6901026 0.83 S1PR1 (0.46) S1PR1CTSSCTSK
SCHEMBL16358672 0.82 S1PR1 (0.40) S1PR1S1PR4THRATHRBRXRA
SCHEMBL3451748 0.81 RXRA (0.50) KDM4ES1PR1HTR2AHTR2CESR1
SCHEMBL16302614 0.81 ALDH1A1 (0.44) KDM4ES1PR1THRBRXRARXRB
Water SCHEMBL27797208 0.81 CTSS (0.51) S1PR1S1PR4THRATHRBCTSS
SCHEMBL2146473 0.80 S1PR4 (0.51) KDM4ES1PR1HTR2AHTR2CS1PR4
SCHEMBL16358671 0.80 S1PR1 (0.38) S1PR1S1PR4THRATHRBRXRA
SCHEMBL13390260 0.79 RXRA (0.50) S1PR1HTR2ARXRARXRBRXRG
SCHEMBL20372428 0.78 PPARD (0.42) S1PR1HTR2CS1PR4RXRARXRB
SCHEMBL16302578 0.77 AAK1 (0.36) KDM4ES1PR1S1PR4THRBRXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011086125-A1 1H-[1,2,3]TRIAZOLO[4,5-c]PYRIDINE-4-CARBONITRILE DERIVATIVES N.V. ORGANON (NL) 2011-07-21 WO disclosed