SCHEMBL6901171

SCHEMBL6901171

NC(=O)OCc1c(F)cccc1F

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 3/20 0.53
MMP2 P08253 3/20 0.53
MMP9 P14780 2/20 0.53
MMP12 P39900 2/20 0.53
NQO1 P15559 1/20 0.44
ALDH1A1 P00352 2/20 0.43
TDP1 Q9NUW8 1/20 0.42
GAA P10253 1/20 0.41
CA5A P35218 1/20 0.41
CES2 O00748 1/20 0.40
CES1 P23141 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
KDM4E B2RXH2 1/20 0.40
MAPT P10636 1/20 0.39
MAOB P27338 1/20 0.39
PARP15 Q460N3 1/20 0.39
PARP14 Q460N5 1/20 0.39
PARP10 Q53GL7 1/20 0.39
CYP1A2 P05177 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27803787 0.89 MMP1 (0.44) MMP1MMP2MMP9MMP12NQO1
SCHEMBL28335441 0.86 ALDH1A1 (0.44) MMP1MMP2MMP9MMP12NQO1
SCHEMBL28686546 0.85 SMN1; SMN2 (0.46) MMP1MMP2MMP9MMP12ALDH1A1
SCHEMBL28724573 0.85 CD38 (0.41) MMP1MMP2MMP9MMP12NQO1
SCHEMBL28740434 0.82 MMP1 (0.40) MMP1MMP2MMP9MMP12NQO1
SCHEMBL28740447 0.81 NQO1 (0.42) MMP1MMP2MMP9MMP12NQO1
SCHEMBL25238748 0.80 MMP1 (0.49) MMP1MMP2MMP9MMP12NQO1
SCHEMBL7630628 0.80 MMP1 (0.53) MMP1MMP2MMP9MMP12ALDH1A1
SCHEMBL22917350 0.80 MMP1 (0.53) MMP1MMP2MMP9MMP12ALDH1A1
SCHEMBL5766366 0.78 ALDH1A1 (0.64) MMP1MMP2MMP9MMP12ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115260211-B Thiophene condensed ring derivative, pharmaceutical composition, preparation method and application thereof 长春金赛药业有限责任公司 2024-02-06 CN disclosed
CN-115260211-A Thiophene fused ring containing derivative, pharmaceutical composition, preparation method and application thereof 长春金赛药业有限责任公司 2022-11-01 CN disclosed
CN-111925379-B Nitrogen-containing heteroaryl substituted pyrimidinediones and uses thereof 广东东阳光药业有限公司 2022-02-15 CN disclosed
CN-111793078-B Bicyclic nitrogen-containing heteroaryl substituted pyrimidinediones and application thereof 东莞市东阳光新药研发有限公司 2022-02-01 CN disclosed
CN-111925379-A Nitrogen-containing heteroaryl substituted pyrimidinediones and uses thereof 广东东阳光药业有限公司 2020-11-13 CN disclosed
CN-111793078-A Bicyclic nitrogen-containing heteroaryl substituted pyrimidinediones and application thereof 东莞市东阳光新药研发有限公司 2020-10-20 CN disclosed
WO-2011060321-A1 TRANSGLUTAMINASE TG2 INHIBITORS, PHARMACEUTICAL COMPOSITIONS, AND METHODS OF USE THEREOF CHDI, INC. (US) 2011-05-19 WO disclosed