SCHEMBL6901717

SCHEMBL6901717

N=C(N)NCCC[C@H](C(N)=O)N(Cc1ccc(CNC(N)=O)cc1)C(=O)C(c1ccc(OCC(=O)O)cc1)c1ccc(OCC(=O)O)cc1

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
EPOR P19235 13/20 0.35
EPHX2 P34913 1/20 0.35
NR1H4 Q96RI1 1/20 0.35
NPY1R P25929 2/20 0.34
NPY4R P50391 2/20 0.34
NPY5R Q15761 1/20 0.34
ITGB3 P05106 1/20 0.34
ITGA2B P08514 1/20 0.34
ALDH1A1 P00352 1/20 0.31
TSHR P16473 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7036782 0.93 EPOR (0.36) EPOREPHX2NR1H4NPY1RNPY4R
SCHEMBL6901908 0.92 KMT2A (0.34) EPORNPY1RNPY4RNPY5RALDH1A1
SCHEMBL8528025 0.89 NPY4R (0.34) EPORNPY1RNPY4RNPY5R
SCHEMBL6900020 0.89 CASR (0.38) ITGB3ITGA2BALDH1A1TSHR
SCHEMBL7043493 0.88 MEN1 (0.35) EPOREPHX2NR1H4NPY1RNPY4R
SCHEMBL7059809 0.88 NPY1R (0.42) NPY1RNPY4RNPY5R
SCHEMBL6899868 0.88 NPY1R (0.42) NPY1RNPY4RNPY5R
SCHEMBL6898240 0.87 NPY1R (0.38) NPY1RNPY4RNPY5R
SCHEMBL6898966 0.86 TDP1 (0.36) NPY1RNPY4RNPY5RTSHR
SCHEMBL6898666 0.86 CYP2C9 (0.45) NPY1RNPY4RNPY5R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0885186-B1 AMINO ACID DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS AND PROCESSES FOR PREPARING THEM THOMAE GMBH DR K (DE) 2003-03-26 EP claimed
US-20040029953-A1 Use of neuropeptide-y antagonists in treatment of alcoholism THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2004-02-12 US disclosed
EP-0885186-B1 AMINO ACID DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS AND PROCESSES FOR PREPARING THEM THOMAE GMBH DR K (DE) 2003-03-26 EP disclosed