SCHEMBL690227

SCHEMBL690227

COc1c(N)cc(C(C)(C)C)cc1CN1CCCC(N(C)C)C1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.44
GAA P10253 1/20 0.44
XBP1 P17861 1/20 0.44
MAPK1 P28482 1/20 0.44
HTT P42858 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
FGFR1 P11362 3/20 0.41
MEN1 O00255 5/20 0.36
KMT2A Q03164 5/20 0.36
POLB P06746 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
DDR1 Q08345 4/20 0.35
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL690226 0.85 ALDH1A1 (0.43) ALDH1A1GAAXBP1MAPK1HTT
SCHEMBL5118355 0.82 CACNA1B (0.43) ALDH1A1GAAXBP1MAPK1HTT
SCHEMBL5124007 0.74 SMN1; SMN2 (0.40) HTTL3MBTL1
SCHEMBL5119240 0.74 KDM4E (0.43) ALDH1A1GAAMEN1KMT2APOLB
SCHEMBL689686 0.71 SSTR5 (0.42) ALDH1A1GAAXBP1MAPK1HTT
SCHEMBL10104443 0.69 ALDH1A1 (0.47) ALDH1A1GAAXBP1MAPK1HTT
SCHEMBL24566256 0.69 MAP4K4 (0.39) FGFR1L3MBTL1DDR1
SCHEMBL24566865 0.69 MAP4K4 (0.39) FGFR1L3MBTL1DDR1
SCHEMBL1935976 0.69 CYP2C19 (0.53) ALDH1A1GAAMAPK1HTTMEN1
SCHEMBL10104438 0.68 ALDH1A1 (0.49) ALDH1A1GAAXBP1MAPK1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2323980-B1 7-(PIPERAZINE-1-YMETHYL)-1H-INDOLE-2-CARBOXYLIC ACID (PHENYL)-AMIDE DERIVATIVES AND ALLIED COMPOUNDS AS P38 MAP KINASE INHIBITORS FOR THE TREATMENT OF RESPIRATORY DISEASES BOEHRINGER INGELHEIM INT (DE) 2012-02-29 EP claimed