SCHEMBL6902319

SCHEMBL6902319

O=C[C@@H]1CN(Cc2ccccc2)C[C@H]1c1ccc(F)c(F)c1

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 2/20 0.42
RORC P51449 2/20 0.41
SIGMAR1 Q99720 2/20 0.41
KDM1A O60341 3/20 0.41
DRD2 P14416 2/20 0.40
DRD3 P35462 2/20 0.40
DPP4 P27487 1/20 0.40
GRIN2B Q13224 1/20 0.39
POLB P06746 1/20 0.39
FUCA1 P04066 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3646250 1.00 CCR5 (0.42) CCR5RORCSIGMAR1KDM1ADRD2
SCHEMBL1713447 1.00 CCR5 (0.42) CCR5RORCSIGMAR1KDM1ADRD2
SCHEMBL6904062 0.90 DRD4 (0.41) CCR5RORCSIGMAR1DRD2DRD3
SCHEMBL1713669 0.88 CCR5 (0.42) CCR5RORCSIGMAR1KDM1ADRD2
SCHEMBL3646393 0.88 CCR5 (0.42) CCR5RORCSIGMAR1KDM1ADRD2
SCHEMBL5274170 0.85 CCR5 (0.57) CCR5RORCSIGMAR1DRD2DRD3
SCHEMBL5236286 0.85 CCR5 (0.57) CCR5RORCSIGMAR1DRD2DRD3
SCHEMBL7827978 0.84 CCR5 (0.50) CCR5RORCSIGMAR1KDM1ADRD2
SCHEMBL5266055 0.84 CCR5 (0.50) CCR5RORCSIGMAR1KDM1ADRD2
SCHEMBL14224261 0.84 CCR5 (0.50) CCR5RORCSIGMAR1KDM1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011073160-A1 PYRROLIDINE DERIVATIVES AS NK - 3 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2011-06-23 WO disclosed