SCHEMBL6904062

SCHEMBL6904062

O=C[C@@H]1CN(Cc2ccccc2)C[C@H]1c1ccc(Cl)c(F)c1

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 1/20 0.41
DPP4 P27487 1/20 0.41
CCR5 P51681 3/20 0.40
RORC P51449 3/20 0.40
DRD2 P14416 2/20 0.39
DRD3 P35462 2/20 0.39
SIGMAR1 Q99720 1/20 0.38
SLC6A2 P23975 1/20 0.38
SLC6A4 P31645 1/20 0.38
SLC6A3 Q01959 1/20 0.38
GRIN2B Q13224 1/20 0.38
FUCA1 P04066 2/20 0.37
CXCR3 P49682 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6902319 0.90 CCR5 (0.42) DPP4CCR5RORCDRD2DRD3
SCHEMBL1713447 0.90 CCR5 (0.42) DPP4CCR5RORCDRD2DRD3
SCHEMBL3646250 0.90 CCR5 (0.42) DPP4CCR5RORCDRD2DRD3
SCHEMBL1713769 0.89 SIGMAR1 (0.47) DRD4DPP4CCR5RORCDRD2
SCHEMBL1714572 0.89 SIGMAR1 (0.47) DRD4DPP4CCR5RORCDRD2
SCHEMBL1507479 0.84 RORC (0.46) DRD4DPP4CCR5RORCDRD2
SCHEMBL5274170 0.83 CCR5 (0.57) CCR5RORCDRD2DRD3SIGMAR1
SCHEMBL5236286 0.83 CCR5 (0.57) CCR5RORCDRD2DRD3SIGMAR1
SCHEMBL7827978 0.82 CCR5 (0.50) DPP4CCR5RORCDRD2DRD3
SCHEMBL5266055 0.82 CCR5 (0.50) DPP4CCR5RORCDRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011073160-A1 PYRROLIDINE DERIVATIVES AS NK - 3 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2011-06-23 WO disclosed