SCHEMBL6904955

SCHEMBL6904955

Cc1ccccc1-c1ccc2nc3c(cc2c1)CC(c1cc(CC(C)(C)C)ncn1)N3

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LCK P06239 1/20 0.38
KDR P35968 1/20 0.38
JAK3 P52333 1/20 0.38
MAPK14 Q16539 1/20 0.38
BACE1 P56817 8/20 0.36
CTSD P07339 2/20 0.36
CLK4 Q9HAZ1 8/20 0.36
CYP1A2 P05177 7/20 0.36
CYP3A4 P08684 7/20 0.36
TSHR P16473 7/20 0.36
CYP2C19 P33261 7/20 0.36
CYP2D6 P10635 5/20 0.36
USP2 O75604 3/20 0.36
LMNA P02545 2/20 0.36
ALDH1A1 P00352 5/20 0.35
MAPK1 P28482 4/20 0.35
HIF1A Q16665 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
CYP2C9 P11712 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1768100 0.71 BACE1 (0.41) LCKKDRJAK3MAPK14BACE1
SCHEMBL1767842 0.68 BACE1 (0.54) LCKKDRJAK3MAPK14BACE1
SCHEMBL1767821 0.68 BACE1 (0.40) LCKKDRJAK3MAPK14BACE1
SCHEMBL14273 0.62 BACE1 (0.41) LCKKDRJAK3MAPK14BACE1
SCHEMBL1767863 0.61 BACE1 (0.55) LCKKDRJAK3MAPK14BACE1
SCHEMBL5491478 0.59 LCK (0.69) LCKKDRJAK3MAPK14BACE1
SCHEMBL1767758 0.57 BACE1 (0.57) LCKKDRJAK3MAPK14BACE1
SCHEMBL24079158 0.57 TGFBR1 (0.40) LCKKDRJAK3MAPK14BACE1
SCHEMBL5157768 0.57 CTSD (0.60) LCKKDRJAK3MAPK14BACE1
SCHEMBL28177941 0.57 BACE1 (0.56) LCKKDRJAK3MAPK14BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011063272-A1 AMINO HETEROARYL COMPOUNDS AS BETA-SECRETASE MODULATORS AND METHODS OF USE AMGEN INC. (US) 2011-05-26 WO disclosed