SCHEMBL690870

SCHEMBL690870

NC(=O)OC(=O)CCC(N)C(=O)OC(N)=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 2/20 0.39
BLM P54132 1/20 0.39
PMP22 Q01453 1/20 0.39
KMT2A Q03164 1/20 0.39
SLC1A1 P43005 2/20 0.35
GRM8 O00222 1/20 0.35
GRM6 O15303 1/20 0.35
GRIN2D O15399 1/20 0.35
GRIN3B O60391 1/20 0.35
GSR P00390 1/20 0.35
CYP1A2 P05177 1/20 0.35
GRIK1 P39086 1/20 0.35
GRM5 P41594 1/20 0.35
GRIA1 P42261 1/20 0.35
GRIA2 P42262 1/20 0.35
GRIA3 P42263 1/20 0.35
SLC1A3 P43003 1/20 0.35
SLC1A2 P43004 1/20 0.35
GRIA4 P48058 1/20 0.35
GRIN1 Q05586 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL690871 1.00 ALOX15 (0.39) ALOX15BLMPMP22KMT2ASLC1A1
SCHEMBL8652131 0.83 KMT2A (0.59) ALOX15BLMPMP22KMT2ASLC1A1
SCHEMBL8648790 0.83 KMT2A (0.59) ALOX15BLMPMP22KMT2ASLC1A1
SCHEMBL20568580 0.83 GRM8 (0.56) ALOX15BLMPMP22KMT2ASLC1A1
SCHEMBL690872 0.83 GRM8 (0.56) ALOX15BLMPMP22KMT2ASLC1A1
SCHEMBL352342 0.82 ALOX15 (0.52) ALOX15BLMPMP22KMT2ASLC1A1
SCHEMBL28571398 0.82 ALOX15 (0.52) ALOX15BLMPMP22KMT2ASLC1A1
SCHEMBL3762162 0.79 SLC1A1 (0.40) ALOX15BLMPMP22KMT2ASLC1A1
SCHEMBL435288 0.79 SLC1A1 (0.40) ALOX15BLMPMP22KMT2ASLC1A1
SCHEMBL5187828 0.79 ALOX15 (0.39) ALOX15BLMPMP22KMT2ASLC1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2421954-B1 DIFFERENTIATED HUMAN LIVER CELL CULTURES AND THEIR USE IN BIOARTIFICIAL LIVER SYSTEMS ACADEMISCH ZIEKENHUIS BIJ DE UNIV VAN AMSTERDAM (NL) 2018-12-26 EP claimed
US-20150073389-A1 DIFFERENTIATED HUMAN LIVER CELL CULTURES AND THEIR USE IN BIOARTIFICIAL LIVER SYSTEMS ACADEMISCH ZIEKENHUIS BIJ DE UNIVERSITEIT VAN AMSTERDAM (NL) 2015-03-12 US claimed
US-8921108-B2 Differentiated human liver cell cultures and their use in bioartificial liver systems ACADEMISCH ZIEKENHUIS BIJ DE UNIVERSITEIT VAN AMSTERDAM (NL) 2014-12-30 US claimed
US-20120111795-A1 DIFFERENTIATED HUMAN LIVER CELL CULTURES AND THEIR USE IN BIOARTIFICIAL LIVER SYSTEMS ACADEMISCH ZIEKENHUIS BIJ DE UNIVERSITEIT VAN AMSTERDAM (NL) 2012-05-10 US claimed
EP-2421954-A1 DIFFERENTIATED HUMAN LIVER CELL CULTURES AND THEIR USE IN BIOARTIFICIAL LIVER SYSTEMS Academisch Ziekenhuis bij de Universiteit van Amsterdam (NL) 2012-02-29 EP claimed
WO-2010123357-A1 DIFFERENTIATED HUMAN LIVER CELL CULTURES AND THEIR USE IN BIOARTIFICIAL LIVER SYSTEMS ACADEMISCH ZIEKENHUIS BIJ DE UNIVERSITEIT VAN AMSTERDAM (NL) 2010-10-28 WO claimed
EP-2421954-B1 DIFFERENTIATED HUMAN LIVER CELL CULTURES AND THEIR USE IN BIOARTIFICIAL LIVER SYSTEMS ACADEMISCH ZIEKENHUIS BIJ DE UNIV VAN AMSTERDAM (NL) 2018-12-26 EP disclosed
US-20150073389-A1 DIFFERENTIATED HUMAN LIVER CELL CULTURES AND THEIR USE IN BIOARTIFICIAL LIVER SYSTEMS ACADEMISCH ZIEKENHUIS BIJ DE UNIVERSITEIT VAN AMSTERDAM (NL) 2015-03-12 US disclosed
US-8921108-B2 Differentiated human liver cell cultures and their use in bioartificial liver systems ACADEMISCH ZIEKENHUIS BIJ DE UNIVERSITEIT VAN AMSTERDAM (NL) 2014-12-30 US disclosed
US-20120111795-A1 DIFFERENTIATED HUMAN LIVER CELL CULTURES AND THEIR USE IN BIOARTIFICIAL LIVER SYSTEMS ACADEMISCH ZIEKENHUIS BIJ DE UNIVERSITEIT VAN AMSTERDAM (NL) 2012-05-10 US disclosed
EP-2421954-A1 DIFFERENTIATED HUMAN LIVER CELL CULTURES AND THEIR USE IN BIOARTIFICIAL LIVER SYSTEMS Academisch Ziekenhuis bij de Universiteit van Amsterdam (NL) 2012-02-29 EP disclosed
WO-2010123357-A1 DIFFERENTIATED HUMAN LIVER CELL CULTURES AND THEIR USE IN BIOARTIFICIAL LIVER SYSTEMS ACADEMISCH ZIEKENHUIS BIJ DE UNIVERSITEIT VAN AMSTERDAM (NL) 2010-10-28 WO disclosed