SCHEMBL6912895

SCHEMBL6912895

C=C(C)c1cccc(CN(CC)Cc2ccc(C(C)(C)C)cc2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
BCHE P06276 3/20 0.40
LTA4H P09960 1/20 0.40
NR1H4 Q96RI1 1/20 0.40
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
ACHE P22303 2/20 0.39
HRH3 Q9Y5N1 1/20 0.39
AOC3 Q16853 1/20 0.39
MEN1 O00255 1/20 0.39
MAPT P10636 1/20 0.39
KMT2A Q03164 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
PPARG P37231 2/20 0.38
KDM4E B2RXH2 1/20 0.38
NR4A1 P22736 1/20 0.37
NR4A2 P43354 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6913077 0.99 ACHE (0.41) HDAC8HDAC6BCHELTA4HNR1H4
SCHEMBL6912986 0.87 HDAC8 (0.47) HDAC8HDAC6BCHELTA4HNR1H4
SCHEMBL6915496 0.86 ACHE (0.49) NR1H4CYP2D6ACHEMEN1MAPT
SCHEMBL610694 0.86 BCHE (0.47) HDAC8HDAC6BCHELTA4HCYP1A2
Hydrochloric Acid SCHEMBL6914315 0.85 SIGMAR1 (0.48) NR1H4CYP2D6ACHEMEN1MAPT
SCHEMBL6914095 0.83 OPRK1 (0.41) HDAC6NR1H4CYP2D6ACHEMEN1
Hydrochloric Acid SCHEMBL6913534 0.82 OPRK1 (0.41) HDAC6NR1H4CYP2D6ACHEMEN1
SCHEMBL6910541 0.81 HDAC3 (0.42) HDAC8HDAC6NR1H4CYP1A2CYP2D6
Hydrochloric Acid SCHEMBL6916238 0.80 HDAC3 (0.41) HDAC8HDAC6NR1H4CYP1A2CYP2D6
SCHEMBL14587216 0.78 CNR2 (0.53) BCHENR1H4CYP1A2CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1112998-B1 AMINE DERIVATIVES POLA CHEM IND INC (JP) 2004-12-08 EP disclosed
US-6586633-B1 Antifungal agents POLA CHEMICAL INDUSTRIES, INC. (JP) 2003-07-01 US disclosed
EP-1112998-A1 AMINE DERIVATIVES POLA CHEMICAL INDUSTRIES, INC. (JP) 2001-07-04 EP disclosed