SCHEMBL6918728

SCHEMBL6918728

C[C@H]1C[C@@H](C(=O)NCc2cc(Cl)ccc2-n2cncn2)N(C(=O)C2(O)c3ccccc3-c3ccccc32)C1

nearest known ligand 0.52

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
F2 P00734 17/20 0.52
PRSS1 P07477 1/20 0.41
CYP3A4 P08684 2/20 0.39
MASP2 O00187 1/20 0.38
CTSL P07711 1/20 0.38
CTSS P25774 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6918723 1.00 F2 (0.52) F2PRSS1CYP3A4MASP2CTSL
SCHEMBL6919843 0.91 F2 (0.53) F2PRSS1
SCHEMBL6078552 0.86 F2 (0.69) F2PRSS1
SCHEMBL6079196 0.75 F2 (0.69) F2PRSS1CYP3A4
SCHEMBL6918158 0.74 ALDH1A1 (0.49) F2PRSS1CYP3A4CTSLCTSS
SCHEMBL6919374 0.72 CYP3A4 (0.54) F2PRSS1CYP3A4
SCHEMBL6919370 0.72 CYP3A4 (0.54) F2PRSS1CYP3A4
SCHEMBL6919773 0.72 F2 (0.40) F2PRSS1CYP3A4CTSLCTSS
SCHEMBL6921244 0.71 F2 (0.47) F2PRSS1CYP3A4
SCHEMBL6919204 0.70 F2 (0.48) F2PRSS1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004032834-A2 THROMBIN INHIBITORS MERCK & CO., INC. (US) 2004-04-22 WO disclosed