SCHEMBL6919140

SCHEMBL6919140

N#CCc1csc(NC(=O)c2ccccc2)n1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.64
PDE5A O76074 2/20 0.64
NPC1 O15118 3/20 0.58
RAB9A P51151 3/20 0.58
CDK5 Q00535 7/20 0.58
CDK5R1 Q15078 7/20 0.58
SMN1; SMN2 Q16637 2/20 0.55
PDE1A P54750 1/20 0.54
PDE1B Q01064 1/20 0.54
PDE1C Q14123 1/20 0.54
AOC3 Q16853 2/20 0.54
KDM4A O75164 1/20 0.53
KDM4B O94953 1/20 0.53
ADORA3 P0DMS8 1/20 0.53
KDM5B Q9UGL1 1/20 0.53
CCNE2 O96020 1/20 0.52
CCNE1 P24864 1/20 0.52
CDK2 P24941 1/20 0.52
SCD O00767 1/20 0.52
MEN1 O00255 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2664522 0.82 KDM4E (0.66) KDM4EPDE5ANPC1RAB9ACDK5
SCHEMBL2664517 0.82 KDM4E (0.69) KDM4EPDE5ANPC1RAB9ACDK5
SCHEMBL27599948 0.82 KDM4E (0.78) KDM4EPDE5ANPC1RAB9ASMN1; SMN2
SCHEMBL2227204 0.82 KDM4E (0.69) KDM4EPDE5ANPC1RAB9ACDK5
SCHEMBL91391 0.82 KDM4E (0.69) KDM4EPDE5ANPC1RAB9ACDK5
SCHEMBL27782868 0.80 AOC3 (0.74) KDM4EPDE5ANPC1RAB9ACDK5
SCHEMBL5717620 0.80 KDM4E (0.74) KDM4EPDE5ANPC1RAB9ACDK5
SCHEMBL3904033 0.79 SMN1; SMN2 (0.65) KDM4ENPC1RAB9ACDK5CDK5R1
SCHEMBL25720785 0.77 PDE5A (0.79) KDM4EPDE5ANPC1RAB9ASMN1; SMN2
SCHEMBL27782870 0.76 SMN1; SMN2 (0.62) KDM4EPDE5ANPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004108722-A1 ORTHOCONDENSED POLYCYCLIC AMINOPYRROLE DERIVATIVES COMPRISING AN ELECTRO-ATTRACTIVE SUBSTITUENT, COMBINATION PRODUCTS OF SAID DERIVATIVES, AND METHOD FOR THE PRODUCTION THEREOF PIERRE FABRE UROLOGIE (FR) 2004-12-16 WO disclosed