SCHEMBL692153

SCHEMBL692153

Nc1ccc2nc(-c3cn[nH]c3N[C@@H]3CCC[C@H]3O)sc2c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ILK Q13418 7/20 0.56
MAPT P10636 5/20 0.43
KDM4E B2RXH2 4/20 0.43
GAA P10253 4/20 0.43
NPC1 O15118 4/20 0.43
RAB9A P51151 4/20 0.43
GLA P06280 3/20 0.43
SMN1; SMN2 Q16637 5/20 0.42
TP53 P04637 2/20 0.42
THRB P10828 2/20 0.42
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
ALDH1A1 P00352 2/20 0.41
PKM P14618 2/20 0.41
HPGD P15428 2/20 0.41
POLB P06746 2/20 0.40
CASP1 P29466 2/20 0.40
CASP7 P55210 2/20 0.40
HSD17B10 Q99714 2/20 0.40
PTBP1 P26599 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL692154 1.00 ILK (0.56) ILKMAPTKDM4EGAANPC1
SCHEMBL687103 0.73 ILK (1.00) ILKMAPTKDM4EGAANPC1
SCHEMBL2163482 0.69 ILK (0.71) ILK
SCHEMBL687417 0.69 ILK (0.71) ILK
SCHEMBL2163486 0.69 ILK (0.71) ILK
SCHEMBL6854931 0.64 MAPT (0.73) ILKMAPTKDM4EGAANPC1
SCHEMBL6854930 0.64 MAPT (0.96) MAPTKDM4EGAANPC1RAB9A
SCHEMBL24134255 0.63 ILK (0.39) ILKCSF1RPDGFRBKITPDGFRA
SCHEMBL23500304 0.63 KCNH2 (0.43) ILKCSF1RPDGFRBKITPDGFRA
SCHEMBL1995933 0.63 MAPT (1.00) MAPTKDM4EGAANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1542997-B1 PYRAZOLYLBENZOTHIAZOLE DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS DERMIRA CANADA INC (CA) 2012-02-29 EP disclosed