SCHEMBL6921941

SCHEMBL6921941

CC1Cn2c(nc3cc(-c4ccc(F)cc4)ccc3c2=O)CO1

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 4/20 0.40
KCNH2 Q12809 1/20 0.40
CACNA2D1 P54289 1/20 0.38
ALDH1A1 P00352 1/20 0.37
RAB9A P51151 3/20 0.37
NPC1 O15118 2/20 0.37
LMNA P02545 1/20 0.37
METAP2 P50579 1/20 0.36
CTSD P07339 6/20 0.36
CYP2D6 P10635 1/20 0.36
CYP3A4 P08684 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15865810 0.86 GRM5 (0.38) GRM2KCNH2ALDH1A1RAB9ANPC1
SCHEMBL6922074 0.81 CACNA2D1 (0.45) CACNA2D1ALDH1A1RAB9ANPC1LMNA
SCHEMBL6921994 0.81 METAP2 (0.40) CACNA2D1RAB9ANPC1METAP2CTSD
SCHEMBL6920768 0.79 GRM5 (0.42)
SCHEMBL6920765 0.78 RAB9A (0.43) GRM2ALDH1A1RAB9ANPC1LMNA
SCHEMBL12039994 0.76 GRM5 (0.38) ALDH1A1RAB9ANPC1LMNA
SCHEMBL6921956 0.75 RAB9A (0.45) ALDH1A1RAB9ANPC1LMNACYP3A4
SCHEMBL12039992 0.73 GRM5 (0.38) ALDH1A1
SCHEMBL6923306 0.73 RAB9A (0.43) GRM2ALDH1A1RAB9ANPC1LMNA
SCHEMBL12059022 0.73 GRM2 (0.39) GRM2ALDH1A1CTSDCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011075699-A2 COMPOUNDS FOR TREATING DISORDERS MEDIATED BY METABOTROPIC GLUTAMATE RECEPTOR 5, AND METHODS OF USE THEREOF SUNOVION PHARMACEUTICALS INC. (US) 2011-06-23 WO disclosed