SCHEMBL692284

SCHEMBL692284

O=C(O)c1cccc(-n2[nH]ccc2=O)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM2B Q8NHM5 1/20 0.56
KDM4C Q9H3R0 1/20 0.56
KMT2A Q03164 6/20 0.49
MEN1 O00255 5/20 0.49
ALDH1A1 P00352 3/20 0.49
KDM4E B2RXH2 3/20 0.49
GAA P10253 3/20 0.49
L3MBTL1 Q9Y468 3/20 0.49
HSD17B10 Q99714 2/20 0.49
HPGD P15428 2/20 0.49
MAPT P10636 2/20 0.49
USP2 O75604 1/20 0.49
MYC P01106 1/20 0.49
POLB P06746 1/20 0.49
HSPA1A P0DMV8 1/20 0.49
ALOX15 P16050 1/20 0.49
NR4A1 P22736 1/20 0.49
PTPN7 P35236 1/20 0.49
RECQL P46063 1/20 0.49
BLM P54132 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
3-Aminobenzoic Acid SCHEMBL11798899 0.86 KDM2B (0.49) KDM2BKDM4CKMT2AMEN1ALDH1A1
SCHEMBL7894742 0.78 ALDH1A1 (0.70) KDM2BKDM4CKMT2AMEN1ALDH1A1
SCHEMBL10948802 0.78 MEN1 (0.49) KMT2AMEN1ALDH1A1GAAHPGD
SCHEMBL1232067 0.77 TSHR (0.48) KDM2BKDM4CKMT2AMEN1ALDH1A1
Phosphine SCHEMBL9466938 0.75 TSHR (0.47) KDM2BKDM4CKMT2AMEN1ALDH1A1
SCHEMBL456557 0.75 ALKBH5 (0.56) KMT2AMEN1ALDH1A1GAAL3MBTL1
SCHEMBL10947683 0.75 FAAH (0.49) KMT2AMEN1ALDH1A1KDM4EGAA
SCHEMBL7463136 0.75 DDB1 (0.45) KDM2BKDM4CKMT2AMEN1ALDH1A1
SCHEMBL9450391 0.73 ALDH1A1 (0.46) KDM2BKDM4CKMT2AMEN1ALDH1A1
SCHEMBL7456550 0.71 MAPT (0.44) KMT2AMEN1ALDH1A1GAAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 41 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2421501-A2 KERATIN DYEING COMPOSITIONS COMPRISING A RADICAL SCAVENGER AND USE THEREOF The Procter & Gamble Company (US) 2012-02-29 EP claimed
WO-2010123863-A2 KERATIN DYEING COMPOSITIONS COMPRISING A RADICAL SCAVENGER AND USE THEREOF THE PROCTER & GAMBLE COMPANY (US) 2010-10-28 WO claimed
EP-4247323-A2 GRANULATED HAIR DYE COMPOSITION Wella Germany GmbH (DE) 2023-09-27 EP disclosed
WO-2022106628-A2 GRANULATED HAIR DYE COMPOSITION WELLA GERMANY GMBH (DE) 2022-05-27 WO disclosed
EP-3512488-A1 HAIR COLOR COMPOSITIONS COMPRISING STABLE VIOLET-BLUE TO BLUE IMIDAZOLIUM DYES Noxell Corporation (US) 2019-07-24 EP disclosed
EP-3512604-A1 STABLE YELLOW IMIDAZOLIUM COMPOUNDS AND METHODS FOR THEIR USE Noxell Corporation (US) 2019-07-24 EP disclosed
WO-2018053027-A1 STABLE YELLOW IMIDAZOLIUM COMPOUNDS AND METHODS FOR THEIR USE NOXELL CORPORATION (US) 2018-03-22 WO disclosed
WO-2018053034-A1 HAIR COLOR COMPOSITIONS COMPRISING STABLE VIOLET-BLUE TO BLUE IMIDAZOLIUM DYES NOXELL CORPORATION (US) 2018-03-22 WO disclosed
WO-2018053096-A1 METHOD OF INCREASING UPTAKE AND WASHFASTNESS OF HAIR HEALTH COMPOUNDS THE PROCTER & GAMBLE COMPANY (US) 2018-03-22 WO disclosed
EP-3271026-A1 METHOD OF COLORING HAIR WITH DIRECT DYE COMPOUNDS Noxell Corporation (US) 2018-01-24 EP disclosed
EP-3271027-A1 COMPOSITIONS FOR DYEING HAIR WITH CATIONIC DIRECT DYES Noxell Corporation (US) 2018-01-24 EP disclosed
WO-2013122990-A1 1-HEXYL-1H-PYRAZOLE-4,5-DIAMINE HEMISULFATE, AND ITS USE IN DYEING COMPOSITIONS THE PROCTER & GAMBLE COMPANY (US) 2013-08-22 WO disclosed
WO-2013105992-A1 OXIDATIVE DYEING COMPOSITIONS COMPRISING AN 1-HEXYL/HEPTYL-4,5-DIAMINOPYRAZOLE AND A PYRIDINE AND DERIVATIVES THEREOF THE PROCTER & GAMBLE COMPANY (US) 2013-07-18 WO disclosed
WO-2013085553-A2 OXIDATIVE DYEING COMPOSITIONS COMPRISING AN 1-HEXYL/HEPTYL-4,5-DIAMINOPYRAZOLE AND A BENZO[1,3]DIOXOL-5-YLAMINE AND DERIVATIVES THEREOF THE PROCTER & GAMBLE COMPANY (US) 2013-06-13 WO disclosed
WO-2013085554-A2 OXIDATIVE DYEING COMPOSITIONS COMPRISING AN 1-HEXYL/HEPTYL-4,5-DIAMINOPYRAZOLE AND A NAPHTHALEN-1-OL AND DERIVATIVES THEREOF THE PROCTER & GAMBLE COMPANY (US) 2013-06-13 WO disclosed
WO-2013058814-A1 OXIDATIVE DYEING COMPOSITIONS COMPRISING AN 1-HEXYL/HEPTYL-4,5-DIAMINOPYRAZOLE AND A BENZENE-1,3-DIOL AND DERIVATIVES THEREOF THE PROCTER & GAMBLE COMPANY (US) 2013-04-25 WO disclosed
WO-2013058815-A1 OXIDATIVE DYEING COMPOSITIONS COMPRISING AN 1-HEXYL/HEPTYL-4,5-DIAMINOPYRAZOLE AND A BENZENE-1,3-DIAMINE AND DERIVATIVES THEREOF THE PROCTER & GAMBLE COMPANY (US) 2013-04-25 WO disclosed
WO-2013058816-A1 OXIDATIVE DYEING COMPOSITIONS COMPRISING AN 1-HEXYL/HEPTYL-4,5-DIAMINOPYRAZOLE AND A 2-AMINOPHENOL AND DERIVATIVES THEREOF THE PROCTER & GAMBLE COMPANY (US) 2013-04-25 WO disclosed
EP-2421501-A2 KERATIN DYEING COMPOSITIONS COMPRISING A RADICAL SCAVENGER AND USE THEREOF The Procter & Gamble Company (US) 2012-02-29 EP disclosed
WO-2010123863-A2 KERATIN DYEING COMPOSITIONS COMPRISING A RADICAL SCAVENGER AND USE THEREOF THE PROCTER & GAMBLE COMPANY (US) 2010-10-28 WO disclosed