SCHEMBL6922877

SCHEMBL6922877

Cn1c2cccc(C(=O)N3CCOCC3)c2c2nc[nH]c(=O)c21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
HTT P42858 1/20 0.43
NPSR1 Q6W5P4 1/20 0.41
TP53 P04637 1/20 0.41
ALDH1A1 P00352 3/20 0.40
USP2 O75604 1/20 0.40
BRD4 O60885 1/20 0.40
TAF1 P21675 1/20 0.40
CECR2 Q9BXF3 1/20 0.40
BRD9 Q9H8M2 1/20 0.40
GAA P10253 1/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
KDM4E B2RXH2 1/20 0.38
HPGD P15428 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38
MAP3K7 O43318 1/20 0.38
FLT3 P36888 1/20 0.38
TAB1 Q15750 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6826311 0.89 MAP3K7 (0.46) HSD17B10ALDH1A1GAAKMT2AKDM4E
SCHEMBL6925074 0.81 IP6K1 (0.40) BRD4
SCHEMBL6826464 0.72 PARP1 (0.50) ALDH1A1BRD4MEN1KMT2A
SCHEMBL6923430 0.69 HTT (0.43) HTTBRD4GAA
SCHEMBL6924211 0.69 KMT2A (0.44) HSD17B10TP53ALDH1A1GAAKMT2A
SCHEMBL6826241 0.69 ABCC1 (0.43) HTTNPSR1ALDH1A1BRD4
SCHEMBL20058392 0.66 ALDH1A1 (0.52) HSD17B10SMN1; SMN2NPSR1TP53ALDH1A1
SCHEMBL7121916 0.65 SMN1; SMN2 (0.77) SMN1; SMN2HTTNPSR1TP53ALDH1A1
SCHEMBL19657112 0.65 HTT (0.47) HSD17B10SMN1; SMN2HTTTP53ALDH1A1
SCHEMBL7361803 0.65 HDAC1 (0.46) HSD17B10SMN1; SMN2HTTNPSR1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004111052-A1 PYRROLOPYRIMIDINE DERIVATIVES AS MODULATORS OF MULTI-DRUG RESISTANCE (MDR) XENOVA LIMITED (GB) 2004-12-23 WO disclosed