SCHEMBL6923430

SCHEMBL6923430

Cn1c2cccc(C#N)c2c2nc[nH]c(=O)c21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.43
PARP1 P09874 6/20 0.38
IP6K1 Q92551 1/20 0.38
IP6K3 Q96PC2 1/20 0.38
IP6K2 Q9UHH9 1/20 0.38
BRD4 O60885 2/20 0.37
MCL1 Q07820 1/20 0.36
MAP2K1 Q02750 2/20 0.35
AURKA O14965 1/20 0.35
DAPK3 O43293 1/20 0.35
JAK2 O60674 1/20 0.35
PRKD3 O94806 1/20 0.35
MAP4K4 O95819 1/20 0.35
PAK4 O96013 1/20 0.35
ABL1 P00519 1/20 0.35
CSF1R P07333 1/20 0.35
RET P07949 1/20 0.35
IGF1R P08069 1/20 0.35
MET P08581 1/20 0.35
PDGFRB P09619 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6826464 0.80 PARP1 (0.50) PARP1IP6K1BRD4MAP2K1AURKA
SCHEMBL6924489 0.80 ABCC1 (0.41) HTTIP6K1IP6K3IP6K2BRD4
SCHEMBL6925074 0.77 IP6K1 (0.40) PARP1IP6K1BRD4MAP2K1AURKA
SCHEMBL6826241 0.76 ABCC1 (0.43) HTTPARP1IP6K1BRD4
SCHEMBL6922477 0.75 GAA (0.35) PARP1MAP2K1AURKAJAK2PRKD3
SCHEMBL6826311 0.71 MAP3K7 (0.46) PARP1GAA
SCHEMBL18030917 0.70 IMPDH2 (0.46) HTTMAP2K1GAA
SCHEMBL6819044 0.70 HTT (0.54) HTTPARP1IP6K1IP6K3IP6K2
SCHEMBL6924053 0.69 PARP1 (0.40) PARP1IP6K1IP6K3IP6K2MCL1
SCHEMBL6922877 0.69 HSD17B10 (0.43) HTTBRD4GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004111052-A1 PYRROLOPYRIMIDINE DERIVATIVES AS MODULATORS OF MULTI-DRUG RESISTANCE (MDR) XENOVA LIMITED (GB) 2004-12-23 WO disclosed