SCHEMBL6924151

SCHEMBL6924151

O=Cc1ccc(NCc2ccccc2-c2ccccc2)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 1/20 0.58
FFAR4 Q5NUL3 1/20 0.58
GCG P01275 1/20 0.44
HDAC3 O15379 2/20 0.44
HDAC1 Q13547 2/20 0.44
HDAC2 Q92769 2/20 0.44
HDAC6 Q9UBN7 2/20 0.44
ALDH1A1 P00352 2/20 0.42
ELANE P08246 1/20 0.42
BRD4 O60885 1/20 0.41
BRD9 Q9H8M2 1/20 0.41
DRD1 P21728 2/20 0.41
DRD2 P14416 1/20 0.41
DRD4 P21917 1/20 0.41
DRD5 P21918 1/20 0.41
DRD3 P35462 1/20 0.41
CYP11B1 P15538 1/20 0.41
CYP11B2 P19099 1/20 0.41
DPP4 P27487 1/20 0.41
APP P05067 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10686619 0.79 MAPT (0.44) ALDH1A1APPHIF1ACYP2A6KMT2A
SCHEMBL6780133 0.79 MEN1 (0.60) FFAR1FFAR4GCGHDAC3HDAC1
SCHEMBL14044097 0.78 FFAR1 (0.66) FFAR1FFAR4GCGHDAC3HDAC1
SCHEMBL10692338 0.78 MAPT (0.46) ALDH1A1ELANEBRD4BRD9APP
SCHEMBL511052 0.76 HTT (0.58) FFAR1FFAR4ALDH1A1ELANEHIF1A
SCHEMBL6237822 0.76 FFAR1 (0.75) FFAR1FFAR4GCGHDAC3HDAC1
SCHEMBL6779496 0.76 FFAR1 (0.55) FFAR1FFAR4GCGHDAC3HDAC1
SCHEMBL9843362 0.76 MAPT (0.43) FFAR1FFAR4DRD1DRD2DRD4
SCHEMBL6778391 0.75 FFAR1 (0.55) FFAR1FFAR4ALDH1A1HIF1AKMT2A
SCHEMBL28660124 0.74 GAA (0.46) HDAC3HDAC1HDAC2HDAC6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6518268-B1 Telomerase inhibitors and methods of their use GERON CORPORATION 2003-02-11 US disclosed
WO-2001002377-A9 TELOMERASE INHIBITORS AND METHODS OF THEIR USE GERON CORP (US) 2001-10-11 WO disclosed
EP-1109796-A1 TELOMERASE INHIBITORS AND METHODS OF THEIR USE Geron Corporation (US) 2001-06-27 EP disclosed
WO-2001002377-A1 TELOMERASE INHIBITORS AND METHODS OF THEIR USE GERON CORPORATION (US) 2001-01-11 WO disclosed