SCHEMBL6924358

SCHEMBL6924358

C[C@@H]1CN([C@H](c2ccc(C#N)cc2)c2cccc(O)c2)[C@@H](C)CN1

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
HPGD P15428 1/20 0.40
OPRM1 P35372 1/20 0.40
OPRK1 P41145 1/20 0.40
SIGMAR1 Q99720 1/20 0.40
ESR1 P03372 1/20 0.39
ESR2 Q92731 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6935200 0.87 SIGMAR1 (0.43) OPRD1CYP1A2CYP3A4CYP2C9HPGD
SCHEMBL6932627 0.87 SIGMAR1 (0.43) OPRD1CYP1A2CYP3A4CYP2C9HPGD
SCHEMBL6932624 0.87 SIGMAR1 (0.43) OPRD1CYP1A2CYP3A4CYP2C9HPGD
SCHEMBL2750726 0.82 OPRD1 (0.51) OPRD1CYP1A2CYP3A4CYP2C9HPGD
SCHEMBL2751375 0.82 OPRD1 (0.51) OPRD1CYP1A2CYP3A4CYP2C9HPGD
SCHEMBL21831852 0.81 DGKA (0.46) OPRD1SIGMAR1
SCHEMBL6925678 0.80 CYP1A2 (0.47) OPRD1CYP1A2CYP3A4CYP2C9HPGD
SCHEMBL6928895 0.79 OPRD1 (0.33) OPRD1CYP1A2CYP3A4OPRM1
SCHEMBL6472695 0.79 CYP1A2 (0.42) OPRD1CYP1A2CYP3A4CYP2C9HPGD
SCHEMBL7623057 0.79 CYP1A2 (0.37) OPRD1CYP1A2CYP3A4CYP2C9HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6514975-B1 Tetrazoles as selective agonists for the delta opioid receptor PFIZER INC 2003-02-04 US disclosed