SCHEMBL6924635

SCHEMBL6924635

CC(c1cccc2ccccc12)N1C(=O)c2c(F)c(F)c(F)c(F)c2C1=O

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ANPEP P15144 2/20 0.45
DPP4 P27487 2/20 0.45
HSD11B1 P28845 2/20 0.40
ALDH1A1 P00352 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
USP2 O75604 1/20 0.38
NPBWR1 P48145 1/20 0.37
PDE2A O00408 1/20 0.36
XIAP P98170 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6924631 1.00 ANPEP (0.45) ANPEPDPP4HSD11B1ALDH1A1CYP1A2
SCHEMBL6921473 1.00 ANPEP (0.45) ANPEPDPP4HSD11B1ALDH1A1CYP1A2
SCHEMBL6923507 0.81 POLB (0.49) DPP4HSD11B1ALDH1A1CYP1A2CYP2C9
SCHEMBL6923510 0.81 POLB (0.49) DPP4HSD11B1ALDH1A1CYP1A2CYP2C9
SCHEMBL23417537 0.79 HSD11B1 (0.41) HSD11B1ALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL13878064 0.79 HSD11B1 (0.41) HSD11B1ALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL23417534 0.79 HSD11B1 (0.41) HSD11B1ALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL719504 0.76 HSD11B1 (0.47) HSD11B1ALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL6919908 0.74 ALDH1A1 (0.44) ANPEPDPP4ALDH1A1
SCHEMBL6919906 0.74 ALDH1A1 (0.44) ANPEPDPP4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6515129-B1 A pharmaceutical composition which comprises, a cyclic imide derivative represented by the general formula (I): present invention relates to an aminopeptidase N inhibitor or an angiogenesis inhibitor, modulates production of tumor necrosis ISHIHARA SANGYO KAISHA LTD. (JP) 2003-02-04 US disclosed
US-6429212-B1 AMINOPEPTIDASE N INHIBITOR USED TO TREAT CANCER, TUMORS, AND RETINOPATHY; FEW SIDE EFFECTS; ANGIOGENESIS INHIBITOR ISHIHARA SANGYO KAISHA LTD. (JP) 2002-08-06 US disclosed