SCHEMBL6924700

SCHEMBL6924700

COc1ccccc1N1CCN(C(=O)CCc2c[nH]c3ccccc23)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 1.00
LMNA P02545 3/20 1.00
MEN1 O00255 2/20 1.00
ALDH1A1 P00352 2/20 0.71
GLA P06280 1/20 0.67
KDM4E B2RXH2 1/20 0.64
GAA P10253 1/20 0.64
MAPT P10636 1/20 0.64
SMN1; SMN2 Q16637 1/20 0.64
TACR1 P25103 6/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6928580 0.90 MEN1 (0.82) KMT2ALMNAMEN1ALDH1A1TACR1
SCHEMBL766304 0.83 KMT2A (0.71) KMT2ALMNAMEN1ALDH1A1GLA
SCHEMBL27715387 0.82 MEN1 (0.69) KMT2ALMNAMEN1MAPT
SCHEMBL11825700 0.81 KMT2A (0.85) KMT2ALMNAMEN1ALDH1A1GLA
SCHEMBL11829657 0.80 TACR1 (0.73) KMT2ALMNAMEN1TACR1
SCHEMBL9215143 0.80 KMT2A (0.66) KMT2ALMNAMEN1ALDH1A1GLA
SCHEMBL11820831 0.80 HTR1A (0.79) KMT2ALMNAMEN1
SCHEMBL6929131 0.80 TACR1 (0.72) KMT2ALMNAMEN1TACR1
SCHEMBL2263678 0.79 KMT2A (0.97) KMT2ALMNAMEN1ALDH1A1GLA
SCHEMBL9650859 0.79 KMT2A (0.66) KMT2ALMNAMEN1ALDH1A1GLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6518273-B1 2-aryl indole derivative as antagonists of tachykinins MERCK SHARP & DOHME LTD. 2003-02-11 US disclosed
WO-2000051984-A1 2-ARYL INDOLE DERIVATIVES AS ANTAGONISTS OF TACHYKININS MERCK SHARP & DOHME LIMITED (GB) 2000-09-08 WO disclosed