SCHEMBL6927082

SCHEMBL6927082

Cc1ccc(S(=O)(=O)Nc2ccc(C(=O)Nc3cccc(/C=C4/SC(=O)NC4=O)c3)cc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 1/20 0.51
MAPT P10636 4/20 0.51
HTT P42858 2/20 0.51
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51
RECQL P46063 1/20 0.51
MEN1 O00255 6/20 0.50
KMT2A Q03164 6/20 0.50
LMNA P02545 3/20 0.49
ALDH1A1 P00352 3/20 0.49
HPGD P15428 2/20 0.49
PIM1 P11309 2/20 0.49
PIM2 Q9P1W9 2/20 0.49
SNCA P37840 1/20 0.47
HDAC4 P56524 2/20 0.47
HDAC8 Q9BY41 2/20 0.47
PPARG P37231 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6927087 1.00 NAMPT (0.51) NAMPTMAPTHTTCYP1A2CYP3A4
SCHEMBL6929936 0.92 KMT2A (0.51) MAPTHTTMEN1KMT2ALMNA
SCHEMBL6929933 0.92 KMT2A (0.51) MAPTHTTMEN1KMT2ALMNA
SCHEMBL6927180 0.91 MEN1 (0.52) NAMPTMAPTHTTMEN1KMT2A
SCHEMBL6927181 0.91 MEN1 (0.52) NAMPTMAPTHTTMEN1KMT2A
SCHEMBL6927642 0.91 PSD (0.54) MAPTHTTMEN1KMT2ALMNA
SCHEMBL6927645 0.91 PSD (0.54) MAPTHTTMEN1KMT2ALMNA
SCHEMBL6926923 0.87 PIM1 (0.54) LMNAPIM1PIM2HDAC4HDAC8
SCHEMBL6926921 0.87 PIM1 (0.54) LMNAPIM1PIM2HDAC4HDAC8
SCHEMBL6928923 0.83 PIM1 (0.67) MAPTHTTMEN1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6518268-B1 Telomerase inhibitors and methods of their use GERON CORPORATION 2003-02-11 US disclosed
WO-2001002377-A9 TELOMERASE INHIBITORS AND METHODS OF THEIR USE GERON CORP (US) 2001-10-11 WO disclosed
EP-1109796-A1 TELOMERASE INHIBITORS AND METHODS OF THEIR USE Geron Corporation (US) 2001-06-27 EP disclosed
WO-2001002377-A1 TELOMERASE INHIBITORS AND METHODS OF THEIR USE GERON CORPORATION (US) 2001-01-11 WO disclosed