SCHEMBL6929936

SCHEMBL6929936

O=C1NC(=O)C(=Cc2cccc(NC(=O)c3ccc(NS(=O)(=O)c4ccccc4)cc3)c2)S1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 7/20 0.51
MEN1 O00255 6/20 0.51
PIM1 P11309 4/20 0.47
PIM2 Q9P1W9 4/20 0.47
PIM3 Q86V86 1/20 0.47
GPR27 Q9NS67 1/20 0.47
AKR1B1 P15121 3/20 0.47
EGFR P00533 1/20 0.46
FGFR1 P11362 1/20 0.46
KDR P35968 1/20 0.46
ALDH1A1 P00352 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
LMNA P02545 1/20 0.46
MAPT P10636 1/20 0.46
MAPK1 P28482 1/20 0.46
HTT P42858 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
USP2 O75604 1/20 0.46
PKM P14618 1/20 0.46
HDAC4 P56524 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6929933 1.00 KMT2A (0.51) KMT2AMEN1PIM1PIM2PIM3
SCHEMBL6927181 0.92 MEN1 (0.52) KMT2AMEN1PIM1PIM2GPR27
SCHEMBL6927180 0.92 MEN1 (0.52) KMT2AMEN1PIM1PIM2GPR27
SCHEMBL6927082 0.92 NAMPT (0.51) KMT2AMEN1PIM1PIM2GPR27
SCHEMBL6927087 0.92 NAMPT (0.51) KMT2AMEN1PIM1PIM2GPR27
SCHEMBL6927642 0.89 PSD (0.54) KMT2AMEN1PIM1PIM2AKR1B1
SCHEMBL6927645 0.89 PSD (0.54) KMT2AMEN1PIM1PIM2AKR1B1
SCHEMBL6926923 0.87 PIM1 (0.54) PIM1PIM2SMN1; SMN2LMNAHDAC4
SCHEMBL6926921 0.87 PIM1 (0.54) PIM1PIM2SMN1; SMN2LMNAHDAC4
SCHEMBL6929942 0.87 MEN1 (0.51) KMT2AMEN1PIM1PIM2PIM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6518268-B1 Telomerase inhibitors and methods of their use GERON CORPORATION 2003-02-11 US disclosed
WO-2001002377-A9 TELOMERASE INHIBITORS AND METHODS OF THEIR USE GERON CORP (US) 2001-10-11 WO disclosed
EP-1109796-A1 TELOMERASE INHIBITORS AND METHODS OF THEIR USE Geron Corporation (US) 2001-06-27 EP disclosed
WO-2001002377-A1 TELOMERASE INHIBITORS AND METHODS OF THEIR USE GERON CORPORATION (US) 2001-01-11 WO disclosed