SCHEMBL6933172

SCHEMBL6933172

CN(C)CC1=C(c2cccc(O)c2)CC(CC2CCCCC2)CCC1

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 15/20 0.38
OPRK1 P41145 13/20 0.38
OPRD1 P41143 12/20 0.38
HRH3 Q9Y5N1 1/20 0.35
ESR1 P03372 1/20 0.35
ESR2 Q92731 1/20 0.35
SLC6A4 P31645 4/20 0.35
SLC6A2 P23975 3/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
CHRNB4 P30926 1/20 0.34
CHRNA3 P32297 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7870812 0.99 OPRM1 (0.39) OPRM1OPRK1OPRD1HRH3ESR1
SCHEMBL6934582 0.87 HRH3 (0.36) OPRM1OPRK1OPRD1HRH3SLC6A4
Hydrochloric Acid SCHEMBL7872718 0.86 OPRM1 (0.37) OPRM1OPRK1OPRD1HRH3SLC6A4
SCHEMBL6934469 0.86 OPRM1 (0.41) OPRM1OPRK1OPRD1ESR1ESR2
SCHEMBL6934080 0.85 OPRK1 (0.40) OPRM1OPRK1OPRD1
Hydrochloric Acid SCHEMBL7874351 0.85 OPRM1 (0.42) OPRM1OPRK1OPRD1ESR1ESR2
Hydrochloric Acid SCHEMBL7876987 0.84 OPRK1 (0.41) OPRM1OPRK1OPRD1
SCHEMBL6936855 0.82 OPRK1 (0.43) OPRM1OPRK1OPRD1
Hydrochloric Acid SCHEMBL7874347 0.81 OPRM1 (0.44) OPRM1OPRK1OPRD1
SCHEMBL6934590 0.81 DRD3 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1010689-B1 Substituted cycloheptenes, their preparation and use GRUENENTHAL GMBH (DE) 2003-01-15 EP claimed
EP-1010689-A1 Substituted cycloheptenes, their preparation and use Grünenthal GmbH (DE) 2000-06-21 EP claimed
EP-1010689-B1 Substituted cycloheptenes, their preparation and use GRUENENTHAL GMBH (DE) 2003-01-15 EP disclosed
EP-1010689-A1 Substituted cycloheptenes, their preparation and use Grünenthal GmbH (DE) 2000-06-21 EP disclosed