SCHEMBL6933543

SCHEMBL6933543

CCCc1nc2cccnc2c(=O)[nH]1

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDM4C Q9H3R0 1/20 0.54
PARP1 P09874 3/20 0.51
PDE10A Q9Y233 3/20 0.46
TNKS2 Q9H2K2 1/20 0.45
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
HTT P42858 1/20 0.42
HPGD P15428 1/20 0.42
PARP2 Q9UGN5 1/20 0.41
ADORA3 P0DMS8 1/20 0.40
HCAR2 Q8TDS4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9844319 0.91 PARP1 (0.63) KDM4CPARP1PDE10ATNKS2HCAR2
SCHEMBL7197836 0.90 PARP1 (0.58) KDM4CPARP1PDE10AHCAR2
SCHEMBL20355457 0.82 PDE10A (0.45) PARP1PDE10ATNKS2NPC1RAB9A
SCHEMBL21072816 0.81 KDM4E (0.43) PARP1PDE10ATNKS2NPC1RAB9A
SCHEMBL20339510 0.81 PARP1 (0.66) PARP1PDE10ATNKS2SMN1; SMN2PARP2
SCHEMBL9853629 0.78 KDM4C (0.48) KDM4CPARP1PDE10ANPC1RAB9A
SCHEMBL29431542 0.76 PARP1 (0.82) KDM4CPARP1PDE10ATNKS2NPC1
SCHEMBL5794718 0.76 PARP1 (0.82) KDM4CPARP1PDE10ATNKS2NPC1
SCHEMBL9432425 0.76 KDM4C (0.50) KDM4CPARP1PDE10ATNKS2HTT
SCHEMBL14281531 0.76 PARP1 (0.56) PARP1TNKS2NPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1365806-A2 USE OF NO ACTTIVATORS FOR TREATMENT AND PREVENTION OF GASTROINTESTINAL DISORDERS JOHNS HOPKINS UNIVERSITY (US) 2003-12-03 EP disclosed
WO-2001078781-A9 METHODS FOR PREVENTION AND TREATMENT OF GASTROINTESTINAL DISORDERS UNIV JOHNS HOPKINS (US) 2002-07-25 WO disclosed
WO-2001078781-A2 METHODS FOR PREVENTION AND TREATMENT OF GASTROINTESTINAL DISORDERS JOHNS HOPKINS UNIVERSITY (US) 2001-10-25 WO disclosed