SCHEMBL6934209

SCHEMBL6934209

NC(=S)NS(=O)(=O)c1cccs1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.57
KMT2A Q03164 4/20 0.57
PKM P14618 1/20 0.57
CYP2D6 P10635 1/20 0.53
CYP2C9 P11712 1/20 0.53
CYP2C19 P33261 1/20 0.53
F2 P00734 2/20 0.50
PRSS1 P07477 2/20 0.50
PRSS2 P07478 2/20 0.50
PRSS3 P35030 2/20 0.50
SLC1A3 P43003 1/20 0.48
SLC1A2 P43004 1/20 0.48
SLC1A1 P43005 1/20 0.48
MEN1 O00255 3/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
TSHR P16473 1/20 0.45
GAA P10253 1/20 0.45
BRAF P15056 1/20 0.44
HKDC1 Q2TB90 1/20 0.44
KDM4E B2RXH2 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL731549 0.84 CYP2D6 (0.55) ALDH1A1KMT2APKMCYP2D6CYP2C9
Urea SCHEMBL8693555 0.82 CYP2D6 (0.53) ALDH1A1KMT2APKMCYP2D6CYP2C9
SCHEMBL10718657 0.82 CYP2D6 (0.53) ALDH1A1KMT2APKMCYP2D6CYP2C9
SCHEMBL8692307 0.78 CYP2D6 (0.56) ALDH1A1KMT2APKMCYP2D6CYP2C9
SCHEMBL10752445 0.78 ALDH1A1 (0.56) ALDH1A1KMT2APKMCYP2D6CYP2C9
SCHEMBL14417207 0.76 CYP2D6 (0.55) ALDH1A1KMT2APKMCYP2D6CYP2C9
SCHEMBL10750707 0.76 ALDH1A1 (0.53) ALDH1A1KMT2APKMCYP2D6CYP2C9
SCHEMBL1863910 0.75 CYP2D6 (0.62) ALDH1A1KMT2APKMCYP2D6CYP2C9
SCHEMBL8232303 0.75 CYP2D6 (0.62) ALDH1A1KMT2APKMCYP2D6CYP2C9
SCHEMBL24254325 0.74 CYP2D6 (0.67) ALDH1A1KMT2ACYP2D6CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0729954-B1 Substituted thiophene sulfonyl ureas and thioureas, process for their preparation, their use as medicaments HOECHST AG (DE) 2003-09-03 EP claimed
CN-1071752-C Substituted thiophenesulfonylureas and-thioureas, processes for their preparation, their use as medicament or diagnostic, and medicament containing them HOECHST AG (DE) 2001-09-26 CN claimed
US-5792788-A FOR TREATMENT OF CARDIAC DISORDERS HOECHST AKTIENGESELLSCHAFT (DE) 1998-08-11 US claimed
CN-1134421-A Substituted thiophenesulfonylureas and-thioureas, processes for their preparation, their use as medicament or diagnostic, and medicament containing them HOECHST AG (DE) 1996-10-30 CN claimed
CN-1071752-C Substituted thiophenesulfonylureas and-thioureas, processes for their preparation, their use as medicament or diagnostic, and medicament containing them HOECHST AG (DE) 2001-09-26 CN disclosed
EP-0885216-A1 SUBSTITUTED THIENYL SULPHONYL (THIO) UREAS AS HERBICIDES BAYER AG (DE) 1998-12-23 EP disclosed
US-5792788-A FOR TREATMENT OF CARDIAC DISORDERS HOECHST AKTIENGESELLSCHAFT (DE) 1998-08-11 US disclosed
WO-1997032875-A1 SUBSTITUTED THIENYL SULPHONYL (THIO) UREAS AS HERBICIDES BAYER AKTIENGESELLSCHAFT (DE) 1997-09-12 WO disclosed
CN-1134421-A Substituted thiophenesulfonylureas and-thioureas, processes for their preparation, their use as medicament or diagnostic, and medicament containing them HOECHST AG (DE) 1996-10-30 CN disclosed
US-4639265-A PRE- AND POSTEMERGENCE E. I. DU PONT DE NEMOURS AND COMPANY (US) 1987-01-27 US disclosed
EP-0064804-B1 THIOPHENE HERBICIDES E.I. DU PONT DE NEMOURS AND COMPANY (US) 1986-07-02 EP disclosed
US-4547217-A ESPECIALLY FOR CORN E. I. DU PONT DE NEMOURS AND COMPANY (US) 1985-10-15 US disclosed
US-4441910-A PRE- AND POST-EMERGENCE E. I. DU PONT DE NEMOURS AND COMPANY (US) 1984-04-10 US disclosed
EP-0064804-A2 Thiophene herbicides E.I. DU PONT DE NEMOURS AND COMPANY (US) 1982-11-17 EP disclosed