SCHEMBL6935035

SCHEMBL6935035

CC(C)CC(NC(=O)C(CCN1C(=O)N(C)C(C)(C)C1=O)SC(=O)c1ccccc1)C(=O)O

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MMP9 P14780 9/20 0.46
MMP3 P08254 8/20 0.46
MMP1 P03956 8/20 0.46
MMP2 P08253 3/20 0.46
MMP13 P45452 2/20 0.46
MMP7 P09237 1/20 0.46
MMP14 P50281 1/20 0.46
MME P08473 3/20 0.40
GRN P28799 1/20 0.37
SORT1 Q99523 1/20 0.37
PLA2G7 Q13093 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6935034 1.00 MMP9 (0.46) MMP9MMP3MMP1MMP2MMP13
SCHEMBL14156438 0.86 MMP1 (0.67) MMP9MMP3MMP1MMP2MMP13
SCHEMBL6766456 0.86 MMP1 (0.67) MMP9MMP3MMP1MMP2MMP13
SCHEMBL4820309 0.84 PLA2G7 (0.46) MMP9MMP3MMP1MMP2MMP13
SCHEMBL4820321 0.84 PLA2G7 (0.46) MMP9MMP3MMP1MMP2MMP13
SCHEMBL4824816 0.84 PLA2G7 (0.46) MMP9MMP3MMP1MMP2MMP13
SCHEMBL14156580 0.78 PLA2G7 (0.47) MMP9MMP3MMP1MMP2MMP13
SCHEMBL14163518 0.78 PLA2G7 (0.47) MMP9MMP3MMP1MMP2MMP13
SCHEMBL4787630 0.78 MMP9 (0.70) MMP9MMP3MMP1MMP2MMP13
SCHEMBL6547584 0.78 MMP9 (0.70) MMP9MMP3MMP1MMP2MMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1123410-B1 THE ENZYME-MEDIATED SYNTHESIS OF PEPTIDOMIMETICS DARWIN DISCOVERY LTD (GB) 2003-12-10 EP disclosed
US-6436697-B1 AMIDATION REACTION OF ORGANOYLSULFANYLALKYLCARBOXYL DERIVATIVE WITH PRIMARY AMINE; ENZYME-MEDIATED COUPLING USING THERMOLYSIN OR SUBTILISIN; AMIDATION, DEBLOCKING, DEPROTECTING DARWIN DISCOVERY, LTD. (GB) 2002-08-20 US disclosed