SCHEMBL6936971

SCHEMBL6936971

CCc1cc(Sc2ccc(Br)cc2)c(C(F)(F)F)cc1C(=O)N=C(N)N

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PLAU P00749 1/20 0.40
SLC9A1 P19634 5/20 0.35
KCNH2 Q12809 2/20 0.35
ICAM1 P05362 1/20 0.34
SELE P16581 1/20 0.34
MC4R P32245 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6935256 0.90 SLC9A1 (0.38) SLC9A1KCNH2ICAM1SELE
SCHEMBL6935062 0.90 ICAM1 (0.40) PLAUSLC9A1KCNH2ICAM1SELE
SCHEMBL6935135 0.89 SLC9A1 (0.38) SLC9A1KCNH2ICAM1SELE
SCHEMBL6935064 0.87 SLC9A1 (0.45) PLAUSLC9A1KCNH2
SCHEMBL6937267 0.84 SLC9A1 (0.36) SLC9A1KCNH2
SCHEMBL6935108 0.83 SLC9A1 (0.40) SLC9A1KCNH2ICAM1SELE
SCHEMBL6935163 0.83 SLC6A2 (0.42) SLC9A1
SCHEMBL6932306 0.82 SLC9A1 (0.40) SLC9A1KCNH2CYP3A4CYP2C9CYP2C19
SCHEMBL6935364 0.82 SLC9A1 (0.43) SLC9A1
SCHEMBL8540499 0.80

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0758644-B1 Sulfonyl- or sulfinyl-benzoyl-guanidine derivatives MERCK PATENT GMBH (DE) 2003-10-15 EP disclosed
US-5744641-A Sulfonyl- or sulfinylbenzoylguanidine derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-04-28 US disclosed
EP-0758644-A1 Sulfonyl- or sulfinyl-benzoyl-guanidine derivatives MERCK PATENT GmbH (DE) 1997-02-19 EP disclosed