SCHEMBL6937137

SCHEMBL6937137

CC1(C)CC(O)c2cc(OCc3ccccc3)ccc2O1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNE1 P15382 3/20 0.55
KCNQ1 P51787 3/20 0.55
MAOB P27338 7/20 0.53
TLR3 O15455 1/20 0.53
CA2 P00918 1/20 0.49
CA5A P35218 1/20 0.49
MAOA P21397 2/20 0.48
ALDH1A1 P00352 2/20 0.46
MAPT P10636 1/20 0.46
HTT P42858 1/20 0.46
TAAR1 Q96RJ0 1/20 0.46
HTR2B P41595 1/20 0.45
TMEM97 Q5BJF2 1/20 0.45
SIGMAR1 Q99720 1/20 0.45
HIF1A Q16665 3/20 0.45
GRIN1 Q05586 2/20 0.45
GRIN2B Q13224 2/20 0.45
NPC1 O15118 1/20 0.42
HPGD P15428 1/20 0.42
NFKB1 P19838 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6601951 0.85 MAOB (0.53) KCNE1KCNQ1MAOBCA2CA5A
SCHEMBL8481853 0.81 KCNE1 (0.54) KCNE1KCNQ1MAOBCA2CA5A
SCHEMBL6603299 0.79 KCNE1 (0.54) KCNE1KCNQ1MAOBCA2CA5A
SCHEMBL8481846 0.79 KCNE1 (0.54) KCNE1KCNQ1MAOBCA2CA5A
SCHEMBL8481843 0.79 KCNE1 (0.52) KCNE1KCNQ1MAOBCA2CA5A
SCHEMBL6603457 0.78 KCNE1 (0.66) KCNE1KCNQ1MAOBMAOAALDH1A1
SCHEMBL6602406 0.78 KCNE1 (0.52) KCNE1KCNQ1MAOBCA2CA5A
SCHEMBL6601126 0.78 KCNE1 (0.68) KCNE1KCNQ1MAOBCA2MAOA
SCHEMBL6934369 0.78 KCNE1 (0.61) KCNE1KCNQ1MAOBCA2CA5A
SCHEMBL4011395 0.77 TLR3 (0.42) KCNE1KCNQ1TLR3ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0913396-B1 Sulphonamide substituted benzopyran derivatives, process of preparation, their use as medicines and pharmaceutical compositions containing them AVENTIS PHARMA GMBH (DE) 2003-09-17 EP disclosed
US-6008245-A TREATMENT OF PROPHYLAXIS AND CARDIOVASCULAR DISORDERS, IN PARTICULAR ARRHYTHMIAS, FOR THE TREATMENT OF ULCERS OF THE GASTROINTESTINAL DISORDERS, DIARRHEAL DISEASES HOECHST MARION ROUSSEL DEUTSCHLAND GMBH (DE) 1999-12-28 US disclosed
EP-0913396-A2 Sulphonamide substituted benzopyran derivatives, process of preparation, their use as medicines and pharmaceutical compositions containing them Hoechst Marion Roussel Deutschland GmbH (DE) 1999-05-06 EP disclosed