SCHEMBL6937435

SCHEMBL6937435

O=C(O)c1cc(Cl)cc(Nc2ccccn2)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 1/20 0.51
ITGAV P06756 1/20 0.51
NPC1 O15118 6/20 0.47
RAB9A P51151 6/20 0.47
HCAR3 P49019 1/20 0.47
GRIK1 P39086 1/20 0.46
JAK2 O60674 1/20 0.45
JAK1 P23458 1/20 0.45
TYK2 P29597 1/20 0.45
TPMT P51580 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
PKM P14618 1/20 0.44
ADORA3 P0DMS8 1/20 0.44
PIM1 P11309 1/20 0.44
ADORA2A P29274 1/20 0.44
ADORA2B P29275 1/20 0.44
ADORA1 P30542 1/20 0.44
FLT3 P36888 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28056305 0.83 MEN1 (0.53) ITGB3ITGAVNPC1RAB9AJAK2
SCHEMBL7105114 0.81 NPC1 (0.63) ITGB3ITGAVNPC1RAB9AHCAR3
SCHEMBL30073949 0.81 NPC1 (0.63) ITGB3ITGAVNPC1RAB9AHCAR3
SCHEMBL4872174 0.79 HCAR3 (0.63) NPC1RAB9AHCAR3SMN1; SMN2MEN1
SCHEMBL11566473 0.75 HCAR3 (0.67) HCAR3
SCHEMBL6841330 0.74 RAB9A (0.56) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL18086899 0.74 KDM4C (0.58) NPC1RAB9AJAK2JAK1TYK2
SCHEMBL3957102 0.73 HTR3E (0.58) NPC1MEN1KMT2AGRM4HDAC6
Hydrochloric Acid SCHEMBL12483461 0.73 GAA (0.56) NPC1RAB9AGRIK1JAK2JAK1
SCHEMBL5177040 0.72 KDM4E (0.55) TPMTADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1097127-B1 DIACYLHYDRAZINE DERIVATIVES AS INTEGRIN INHIBITORS MERCK PATENT GMBH (DE) 2003-03-12 EP disclosed
US-6326403-B1 CARDIOVASCULAR DISORDERS MERCK PATENT GESELLSCHAFT MIT (DE) 2001-12-04 US disclosed