SCHEMBL6938174

SCHEMBL6938174

Cc1cn(CC[C@H](O)CO[Si](C)(C)C(C)(C)C)c2ccccc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TK1 P04183 1/20 0.40
PRMT5 O14744 1/20 0.39
KMT2A Q03164 5/20 0.39
MEN1 O00255 4/20 0.39
MAPT P10636 4/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
GAA P10253 2/20 0.36
HDAC1 Q13547 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
HDAC9 Q9UKV0 1/20 0.35
CREBBP Q92793 1/20 0.35
LMNA P02545 2/20 0.34
HPGD P15428 2/20 0.34
HTT P42858 1/20 0.34
KDM4E B2RXH2 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6938178 1.00 TK1 (0.40) TK1PRMT5KMT2AMEN1MAPT
SCHEMBL6940163 0.80 ADRB2 (0.41) TK1KMT2AMEN1MAPTGAA
SCHEMBL6940159 0.80 ADRB2 (0.41) TK1KMT2AMEN1MAPTGAA
SCHEMBL6939460 0.79 HTR2A (0.46) KMT2AMEN1LMNAHPGDKDM4E
SCHEMBL6939466 0.79 HTR2A (0.46) KMT2AMEN1LMNAHPGDKDM4E
SCHEMBL6933500 0.79 CDK4 (0.45) KMT2AMEN1MAPTNPC1RAB9A
SCHEMBL6933502 0.79 CDK4 (0.45) KMT2AMEN1MAPTNPC1RAB9A
SCHEMBL6939120 0.77 MEN1 (0.38) KMT2AMEN1MAPTNPC1RAB9A
SCHEMBL6942595 0.76 MEN1 (0.38) KMT2AMEN1MAPTNPC1RAB9A
SCHEMBL6941805 0.74 TP53 (0.46) PRMT5KMT2AMEN1MAPTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6596738-B1 Inhibiting activity to adenosine deaminase (hereinafter described as ADA) An adenosine deaminase inhibiting agent comprising a compound of the formula (I): FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-07-22 US disclosed