SCHEMBL6939612

SCHEMBL6939612

CS(=O)(=O)N(NC(=O)[C@H](Cc1ccccc1)[C@H](CC=Cc1ccccc1)C(=O)NO)c1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADAM17 P78536 2/20 0.58
MMP2 P08253 11/20 0.38
MMP3 P08254 8/20 0.38
MMP7 P09237 6/20 0.38
MMP1 P03956 7/20 0.37
MMP9 P14780 6/20 0.37
MMP8 P22894 4/20 0.37
MMP13 P45452 3/20 0.37
MMP12 P39900 1/20 0.37
MMP14 P50281 1/20 0.37
PPARG P37231 1/20 0.36
CNR2 P34972 1/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
CTSC P53634 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6940033 0.93 ADAM17 (0.49) ADAM17MMP2MMP9MMP8MMP13
SCHEMBL6940945 0.88 ADAM17 (0.75) ADAM17MMP2MMP3MMP7MMP1
SCHEMBL6939936 0.86 ADAM17 (0.56) ADAM17MMP2MMP7MMP1MMP9
SCHEMBL6944720 0.84 ADAM17 (0.54) ADAM17MMP2MMP3MMP1MMP9
SCHEMBL6943824 0.84 ADAM17 (0.55) ADAM17MMP2MMP3MMP1MMP9
SCHEMBL6939403 0.84 ADAM17 (0.55) ADAM17MMP2MMP3MMP1MMP9
SCHEMBL6945656 0.83 ADAM17 (0.71) ADAM17MMP2MMP3MMP7MMP1
SCHEMBL6943011 0.81 ADAM17 (0.65) ADAM17MMP2MMP3MMP7MMP1
SCHEMBL6940910 0.81 ADAM17 (0.67) ADAM17MMP2MMP3MMP7MMP1
SCHEMBL6944738 0.80 ADAM17 (0.64) ADAM17MMP2MMP3MMP7MMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0993442-B1 HYDRAZINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2003-04-23 EP disclosed
US-6235787-B1 ANTIINFLAMMATORY AGENTS; RHEUMATIC DISEASES; BONE DISORDERS; SKIN DISORDERS; MULTIPLE SCLEROSIS HOFFMANN-LA ROCHE INC. 2001-05-22 US disclosed