SCHEMBL6943824

SCHEMBL6943824

CS(=O)(=O)N(NC(=O)[C@H](CC1CCCC1)[C@H](CC=Cc1ccccc1)C(=O)NO)c1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADAM17 P78536 1/20 0.55
MMP2 P08253 15/20 0.40
MMP1 P03956 14/20 0.40
MMP3 P08254 14/20 0.40
MMP8 P22894 14/20 0.40
MMP13 P45452 14/20 0.40
POLB P06746 1/20 0.37
ALDH1A1 P00352 1/20 0.37
GAA P10253 1/20 0.37
ATM Q13315 1/20 0.34
MMP9 P14780 1/20 0.34
CTSC P53634 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6939403 0.98 ADAM17 (0.55) ADAM17MMP2MMP1MMP3MMP8
SCHEMBL6942478 0.85 ADAM17 (0.41) ADAM17MMP2MMP1MMP3MMP8
SCHEMBL6943846 0.84 ADAM17 (0.40) ADAM17MMP2MMP1MMP3MMP8
SCHEMBL6940945 0.84 ADAM17 (0.75) ADAM17MMP2MMP1MMP3MMP8
SCHEMBL6939612 0.84 ADAM17 (0.58) ADAM17MMP2MMP1MMP3MMP8
SCHEMBL6939936 0.83 ADAM17 (0.56) ADAM17MMP2MMP1MMP13MMP9
SCHEMBL6944720 0.81 ADAM17 (0.54) ADAM17MMP2MMP1MMP3MMP8
SCHEMBL6945656 0.80 ADAM17 (0.71) ADAM17MMP2MMP1MMP3MMP8
SCHEMBL6939485 0.79 ADAM17 (0.75) ADAM17MMP2MMP1MMP3MMP8
SCHEMBL6946042 0.78 ADAM17 (0.74) ADAM17MMP2MMP1MMP3MMP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0993442-B1 HYDRAZINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2003-04-23 EP disclosed
US-6235787-B1 ANTIINFLAMMATORY AGENTS; RHEUMATIC DISEASES; BONE DISORDERS; SKIN DISORDERS; MULTIPLE SCLEROSIS HOFFMANN-LA ROCHE INC. 2001-05-22 US disclosed