SCHEMBL6939728

SCHEMBL6939728

COc1ccc(CC2(O)CCCCC2C(c2ccccc2)N(C)C)cc1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.40
SLC6A4 P31645 5/20 0.40
SLC6A3 Q01959 5/20 0.40
SLC6A2 P23975 4/20 0.40
CCR5 P51681 1/20 0.40
LMNA P02545 1/20 0.40
CNR1 P21554 1/20 0.40
HTR2A P28223 1/20 0.40
HRH1 P35367 1/20 0.40
HRH3 Q9Y5N1 1/20 0.40
TDP1 Q9NUW8 1/20 0.39
KLK7 P49862 1/20 0.39
CASR P41180 1/20 0.38
OPRM1 P35372 2/20 0.37
OPRL1 P41146 2/20 0.37
OPRD1 P41143 1/20 0.37
OPRK1 P41145 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6936762 0.90 SLC6A9 (0.39) SLC6A4SLC6A3LMNAKLK7OPRM1
Hydrochloric Acid SCHEMBL7741182 0.89 OPRL1 (0.39) SLC6A4SLC6A3LMNAKLK7OPRM1
SCHEMBL5164176 0.89 SLC6A2 (0.44) ALDH1A1SLC6A4SLC6A2CCR5LMNA
SCHEMBL6939045 0.88 CCR5 (0.43) SLC6A4SLC6A3SLC6A2CCR5LMNA
SCHEMBL5163369 0.87 CCR5 (0.38) CCR5TDP1
SCHEMBL5846308 0.87 CCR5 (0.38) SLC6A4SLC6A3SLC6A2CCR5OPRM1
Hydrochloric Acid SCHEMBL5847559 0.86 CCR5 (0.37) SLC6A4SLC6A3SLC6A2CCR5LMNA
SCHEMBL6937455 0.85 PSEN1 (0.37) CCR5LMNACNR1HRH1OPRK1
SCHEMBL6936755 0.83 SLC6A2 (0.47) ALDH1A1SLC6A4SLC6A2CCR5LMNA
SCHEMBL5158039 0.83 MEN1 (0.40) LMNAOPRM1OPRL1OPRD1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1043307-B1 3-amino-3-arylpropan-1-ol-derivates, their preparation and their use GRUENENTHAL GMBH (DE) 2003-06-04 EP claimed
US-6410790-B1 ANALGESICS GRUENENTHAL GMBH (DE) 2002-06-25 US claimed
EP-1043307-A2 3-amino-3-arylpropan-1-ol-derivates, their preparation and their use Grünenthal GmbH (DE) 2000-10-11 EP claimed
EP-1043307-B1 3-amino-3-arylpropan-1-ol-derivates, their preparation and their use GRUENENTHAL GMBH (DE) 2003-06-04 EP disclosed
US-6410790-B1 ANALGESICS GRUENENTHAL GMBH (DE) 2002-06-25 US disclosed
EP-1043307-A2 3-amino-3-arylpropan-1-ol-derivates, their preparation and their use Grünenthal GmbH (DE) 2000-10-11 EP disclosed