SCHEMBL5158039

SCHEMBL5158039

COc1ccccc1CC1(O)CCCCC1C(c1ccccc1)N(C)C

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.40
KMT2A Q03164 4/20 0.40
CRHBP P24387 1/20 0.40
CRHR2 Q13324 1/20 0.40
TACR1 P25103 5/20 0.38
SMN1; SMN2 Q16637 1/20 0.37
SIGMAR1 Q99720 1/20 0.36
ATM Q13315 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
LMNA P02545 1/20 0.35
HPGD P15428 1/20 0.35
OPRM1 P35372 1/20 0.34
OPRD1 P41143 1/20 0.34
OPRK1 P41145 1/20 0.34
OPRL1 P41146 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5162314 0.84 CCR5 (0.38) MEN1KMT2ATACR1SIGMAR1
SCHEMBL5164050 0.84 CCR5 (0.38) MEN1KMT2ASMN1; SMN2LMNAOPRM1
Hydrochloric Acid SCHEMBL5846847 0.83 CCR5 (0.37) MEN1KMT2ATACR1SMN1; SMN2SIGMAR1
SCHEMBL6937462 0.83 DPP4 (0.37) TACR1OPRL1
SCHEMBL6936762 0.83 SLC6A9 (0.39) SMN1; SMN2LMNAOPRM1OPRD1OPRK1
SCHEMBL6939728 0.83 ALDH1A1 (0.40) LMNAOPRM1OPRD1OPRK1OPRL1
SCHEMBL6936254 0.82 C3AR1 (0.37) MEN1KMT2ASMN1; SMN2LMNAOPRM1
Hydrochloric Acid SCHEMBL7741182 0.82 OPRL1 (0.39) SMN1; SMN2LMNAOPRM1OPRD1OPRK1
SCHEMBL6939842 0.81 MEN1 (0.37) MEN1KMT2AOPRM1OPRL1
SCHEMBL5164176 0.80 SLC6A2 (0.44) MEN1KMT2ASIGMAR1LMNAOPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1406857-B1 SUBSTITUTED 1-ARYL-BUT-3-ENYLAMINE AND 1-ARYL-BUT-2-ENYLAMINE COMPOUNDS GRUENENTHAL GMBH (DE) 2007-02-21 EP disclosed