SCHEMBL6940964

SCHEMBL6940964

CC(C)C[C@@H](C(=O)NN(c1nc2ccccc2s1)S(C)(=O)=O)[C@H](CC=Cc1ccccc1)C(=O)NOC1CCCCO1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADAM17 P78536 1/20 0.45
CCNA2 P20248 1/20 0.31
CDK2 P24941 1/20 0.31
CCNA1 P78396 1/20 0.31
CDK5 Q00535 1/20 0.31
CDK5R1 Q15078 1/20 0.31
NPC1 O15118 1/20 0.31
TP53 P04637 1/20 0.31
MAPK1 P28482 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
ALDH1A1 P00352 1/20 0.31
KMT2A Q03164 2/20 0.30
MEN1 O00255 1/20 0.30
GAA P10253 1/20 0.30
ATM Q13315 2/20 0.30
KDM4E B2RXH2 1/20 0.30
TDP1 Q9NUW8 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
TGFBR1 P36897 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6947352 0.88 ADAM17 (0.51) ADAM17CCNA2CDK2CCNA1CDK5
SCHEMBL6946888 0.87 ADAM17 (0.48) ADAM17CCNA2CDK2CCNA1CDK5
SCHEMBL6943006 0.87 ADAM17 (0.46) ADAM17TGFBR1
SCHEMBL7937100 0.85 ADAM17 (0.48) ADAM17TGFBR1TSHR
SCHEMBL6942217 0.85 ADAM17 (0.49) ADAM17L3MBTL1TGFBR1
SCHEMBL6945960 0.85 ADAM17 (0.51) ADAM17TGFBR1
SCHEMBL6937788 0.85 ADAM17 (0.51) ADAM17CCNA2CDK2CCNA1CDK5
SCHEMBL6943375 0.85 ADAM17 (0.53) ADAM17CCNA2CDK2CCNA1CDK5
SCHEMBL6942699 0.84 ADAM17 (0.63) ADAM17NPC1TP53RAB9ASMN1; SMN2
SCHEMBL6945855 0.84 ADAM17 (0.48) ADAM17TGFBR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0993442-B1 HYDRAZINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2003-04-23 EP disclosed
US-6235787-B1 ANTIINFLAMMATORY AGENTS; RHEUMATIC DISEASES; BONE DISORDERS; SKIN DISORDERS; MULTIPLE SCLEROSIS HOFFMANN-LA ROCHE INC. 2001-05-22 US disclosed