SCHEMBL6941172

SCHEMBL6941172

O=C(O)CC12CC3CC(CC(C3)O1)C2

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.41
POLB P06746 1/20 0.41
EPHX2 P34913 5/20 0.38
HSD11B1 P28845 3/20 0.38
KDM4E B2RXH2 1/20 0.37
HTT P42858 1/20 0.37
CYP3A4 P08684 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8104799 0.96 ALDH1A1 (0.39) ALDH1A1POLBEPHX2HSD11B1KDM4E
SCHEMBL14859158 0.77 EPHX2 (0.33) ALDH1A1EPHX2
SCHEMBL2482790 0.73 POLB (0.42) ALDH1A1POLBHSD11B1KDM4EHTT
Adamantaneacetic Acid SCHEMBL24688608 0.72 ALDH1A1 (0.62) ALDH1A1POLBHSD11B1CYP3A4CYP2C19
Adamantaneacetic Acid SCHEMBL306081 0.72 ALDH1A1 (0.62) ALDH1A1POLBHSD11B1CYP3A4CYP2C19
Adamantaneacetic Acid SCHEMBL6865701 0.72 ALDH1A1 (0.62) ALDH1A1POLBHSD11B1CYP3A4CYP2C19
SCHEMBL944175 0.71 EPHX2 (0.37) ALDH1A1EPHX2
Adamantaneacetic Acid SCHEMBL4147939 0.70 ALDH1A1 (0.60) ALDH1A1POLBHSD11B1CYP3A4CYP2C19
SCHEMBL8097478 0.67 HSD11B1 (0.48) ALDH1A1POLBHSD11B1KDM4EHTT
SCHEMBL944090 0.67 EPHX2 (0.37) ALDH1A1EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1036058-B1 ADAMANTANE DERIVATIVES ASTRAZENECA UK LTD (GB) 2003-03-12 EP disclosed
US-6242470-B1 RHEUMATIC DISEASES; ANTIARTHRITIC AGENTS, ANTIALLERGENS; IRRITABLE BOWEL SYNDROME; AMIDATION ASTRAZENECA AB (SE) 2001-06-05 US disclosed
EP-1036058-A1 ADAMANTANE DERIVATIVES AstraZeneca UK Limited (GB) 2000-09-20 EP disclosed
WO-1999029660-A1 ADAMANTANE DERIVATIVES ASTRAZENECA UK LIMITED (GB) 1999-06-17 WO disclosed