SCHEMBL6941223

SCHEMBL6941223

Cc1cc(O)ccc1NC(=O)CC12CC3CC(CC(C3)C1)C2

nearest known ligand 0.70

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 8/20 0.70
GPR55 Q9Y2T6 1/20 0.54
CA12 O43570 1/20 0.51
CA9 Q16790 1/20 0.51
EPHX2 P34913 1/20 0.49
ABCB11 O95342 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6939404 0.90 P2RX7 (0.72) P2RX7GPR55ABCB11
SCHEMBL6594387 0.86 P2RX7 (0.61) P2RX7GPR55CA12CA9
SCHEMBL6941699 0.84 P2RX7 (0.70) P2RX7GPR55
SCHEMBL6939157 0.84 P2RX7 (0.82) P2RX7
SCHEMBL6939826 0.83 P2RX7 (0.68) P2RX7GPR55ABCB11
SCHEMBL18992830 0.82 P2RX7 (0.62) P2RX7
SCHEMBL12932448 0.82 P2RX7 (0.75) P2RX7GPR55CA12CA9EPHX2
SCHEMBL6939890 0.82 P2RX7 (0.70) P2RX7GPR55CA12CA9
SCHEMBL6939213 0.79 P2RX7 (0.59) P2RX7GPR55CA12CA9
SCHEMBL7660416 0.78 P2RX7 (0.58) P2RX7GPR55ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1036058-B1 ADAMANTANE DERIVATIVES ASTRAZENECA UK LTD (GB) 2003-03-12 EP claimed
US-6242470-B1 RHEUMATIC DISEASES; ANTIARTHRITIC AGENTS, ANTIALLERGENS; IRRITABLE BOWEL SYNDROME; AMIDATION ASTRAZENECA AB (SE) 2001-06-05 US claimed
EP-1036058-B1 ADAMANTANE DERIVATIVES ASTRAZENECA UK LTD (GB) 2003-03-12 EP disclosed
US-6242470-B1 RHEUMATIC DISEASES; ANTIARTHRITIC AGENTS, ANTIALLERGENS; IRRITABLE BOWEL SYNDROME; AMIDATION ASTRAZENECA AB (SE) 2001-06-05 US disclosed
EP-1036058-A1 ADAMANTANE DERIVATIVES AstraZeneca UK Limited (GB) 2000-09-20 EP disclosed
WO-1999029660-A1 ADAMANTANE DERIVATIVES ASTRAZENECA UK LIMITED (GB) 1999-06-17 WO disclosed