SCHEMBL6941247

SCHEMBL6941247

Cc1ccc(CO)cc1NC(=O)CC12CC3CC(CC(C3)C1)C2

nearest known ligand 0.69

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 8/20 0.69
ABCB11 O95342 1/20 0.54
GPR55 Q9Y2T6 1/20 0.49
MAPK1 P28482 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6939401 0.87 P2RX7 (0.71) P2RX7ABCB11GPR55MAPK1NPSR1
SCHEMBL6939404 0.85 P2RX7 (0.72) P2RX7ABCB11GPR55MAPK1NPSR1
SCHEMBL7071927 0.84 P2RX7 (0.61) P2RX7ABCB11GPR55NPSR1
SCHEMBL6860227 0.81 P2RX7 (1.00) P2RX7ABCB11MAPK1
SCHEMBL6939826 0.81 P2RX7 (0.68) P2RX7ABCB11GPR55
SCHEMBL6941167 0.81 ALDH1A1 (0.61) P2RX7ABCB11NPSR1
SCHEMBL6943104 0.78 P2RX7 (0.76) P2RX7ABCB11MAPK1NPSR1
SCHEMBL6941223 0.77 P2RX7 (0.70) P2RX7ABCB11GPR55
SCHEMBL6939407 0.76 P2RX7 (0.72) P2RX7ABCB11
SCHEMBL7956634 0.76 P2RX7 (0.72) P2RX7ABCB11GPR55MAPK1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1036058-B1 ADAMANTANE DERIVATIVES ASTRAZENECA UK LTD (GB) 2003-03-12 EP claimed
US-6242470-B1 RHEUMATIC DISEASES; ANTIARTHRITIC AGENTS, ANTIALLERGENS; IRRITABLE BOWEL SYNDROME; AMIDATION ASTRAZENECA AB (SE) 2001-06-05 US claimed
EP-1036058-B1 ADAMANTANE DERIVATIVES ASTRAZENECA UK LTD (GB) 2003-03-12 EP disclosed
US-6242470-B1 RHEUMATIC DISEASES; ANTIARTHRITIC AGENTS, ANTIALLERGENS; IRRITABLE BOWEL SYNDROME; AMIDATION ASTRAZENECA AB (SE) 2001-06-05 US disclosed