SCHEMBL6941744

SCHEMBL6941744

c1coc(Cn2cnc3cncnc32)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
STAT3 P40763 1/20 0.52
HDAC1 Q13547 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
HSD17B10 Q99714 5/20 0.46
HPGD P15428 5/20 0.44
FDPS P14324 1/20 0.44
LTA4H P09960 1/20 0.43
HTT P42858 3/20 0.41
NPSR1 Q6W5P4 5/20 0.40
MAPT P10636 4/20 0.40
MEN1 O00255 4/20 0.40
LMNA P02545 4/20 0.40
KMT2A Q03164 4/20 0.40
ALOX15 P16050 3/20 0.40
TP53 P04637 2/20 0.40
TSHR P16473 2/20 0.40
MAPK1 P28482 1/20 0.40
BRCA1 P38398 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
ALDH1A1 P00352 8/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15692 0.77 CCNB2 (0.40) HSD17B10HPGDHTTNPSR1MAPT
9-Benzyl-9H-Purine SCHEMBL434620 0.76 HDAC1 (0.61) HDAC1HDAC6HSD17B10FDPSLTA4H
SCHEMBL526066 0.73 ADORA2A (0.62) HSD17B10HPGDHTTLMNASMN1; SMN2
SCHEMBL10857669 0.73 FDPS (0.54) HDAC1HDAC6HSD17B10FDPSLTA4H
SCHEMBL6948681 0.72 HDAC1 (0.46) HDAC1HDAC6HPGDFDPSLTA4H
SCHEMBL6942099 0.72 MKNK2 (0.40) HDAC1HDAC6HSD17B10FDPSLTA4H
SCHEMBL27932506 0.72 FDPS (0.53) HDAC1HDAC6HSD17B10FDPSLTA4H
SCHEMBL10442248 0.71 PDE4A (0.54) HDAC1HDAC6FDPSLTA4HMEN1
SCHEMBL5493573 0.71 HDAC6 (0.50) HDAC1HDAC6HSD17B10FDPSLTA4H
SCHEMBL6944736 0.71 HDAC1 (0.62) HDAC1HDAC6FDPSLTA4HHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1349857-A1 PURINE DERIVATIVES AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2003-10-08 EP disclosed
WO-2002055521-A1 PURINE DERIVATIVES AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2002-07-18 WO disclosed