SCHEMBL6944736

SCHEMBL6944736

Cc1ccc(Cn2cnc3cncnc32)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.62
HDAC6 Q9UBN7 1/20 0.62
LMNA P02545 4/20 0.54
CYP11B1 P15538 4/20 0.54
CYP11B2 P19099 4/20 0.54
HTT P42858 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
LTA4H P09960 1/20 0.48
FDPS P14324 1/20 0.46
PDE10A Q9Y233 1/20 0.45
CYP1A2 P05177 4/20 0.44
CYP2C19 P33261 4/20 0.44
CYP3A4 P08684 3/20 0.44
USP2 O75604 2/20 0.44
ALDH1A1 P00352 2/20 0.44
TSHR P16473 2/20 0.44
CYP2C9 P11712 3/20 0.43
MEN1 O00255 4/20 0.43
KMT2A Q03164 4/20 0.43
HBB P68871 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
9-Benzyl-9H-Purine SCHEMBL434620 0.84 HDAC1 (0.61) HDAC1HDAC6LMNACYP11B1CYP11B2
SCHEMBL28195658 0.84 HDAC1 (0.58) HDAC1HDAC6LMNACYP11B1CYP11B2
SCHEMBL6946826 0.81 HDAC6 (0.62) HDAC1HDAC6LMNALTA4HFDPS
SCHEMBL12472771 0.79 HDAC6 (0.72) HDAC1HDAC6LMNACYP11B2SMN1; SMN2
SCHEMBL15705713 0.79 HDAC6 (0.80) HDAC1HDAC6LTA4HFDPSMEN1
SCHEMBL30983905 0.77 HDAC1 (0.45) HDAC1HDAC6LMNACYP11B1CYP11B2
SCHEMBL12472812 0.77 HDAC6 (1.00) HDAC1HDAC6FDPSMEN1KMT2A
SCHEMBL6945092 0.77 HDAC6 (0.64) HDAC1HDAC6LMNACYP11B1CYP11B2
SCHEMBL31229302 0.76 CYP11B1 (0.66) LMNACYP11B1CYP11B2HTTSMN1; SMN2
SCHEMBL29914166 0.75 USP1 (0.57) HDAC1HDAC6LTA4HCYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1349857-A1 PURINE DERIVATIVES AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2003-10-08 EP disclosed
WO-2002055521-A1 PURINE DERIVATIVES AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2002-07-18 WO disclosed
CN-1135485-A 2,9-di-substituted pur-6-ones compound BAYER AG (DE) 1996-11-13 CN disclosed