SCHEMBL6943306

SCHEMBL6943306

CC(C)C[C@@H](C(=O)NN(c1ccccc1)S(C)(=O)=O)C(CC=Cc1cccnc1)C(=O)NOC1CCCCO1

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADAM17 P78536 1/20 0.45
CHRNB2 P17787 1/20 0.35
CHRNA4 P43681 1/20 0.35
TGFBR1 P36897 1/20 0.32
MMP1 P03956 1/20 0.32
MMP2 P08253 1/20 0.32
MMP3 P08254 1/20 0.32
MMP7 P09237 1/20 0.32
C3AR1 Q16581 1/20 0.32
GAA P10253 1/20 0.31
P2RX3 P56373 1/20 0.30
POLB P06746 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6947352 0.94 ADAM17 (0.51) ADAM17TGFBR1MMP2GAAP2RX3
SCHEMBL6945960 0.90 ADAM17 (0.51) ADAM17TGFBR1MMP2P2RX3
SCHEMBL6940024 0.88 ADAM17 (0.48) ADAM17MMP1MMP2MMP3POLB
SCHEMBL6942385 0.88 ADAM17 (0.45) ADAM17TGFBR1P2RX3POLB
SCHEMBL6944673 0.87 ADAM17 (0.46) ADAM17MMP1P2RX3
SCHEMBL6942441 0.87 ADAM17 (0.45) ADAM17TGFBR1MMP1P2RX3
SCHEMBL6940527 0.87 ADAM17 (0.46) ADAM17TGFBR1MMP2GAAP2RX3
SCHEMBL6943951 0.86 ADAM17 (0.51) ADAM17CHRNB2CHRNA4TGFBR1MMP1
SCHEMBL6946852 0.86 ADAM17 (0.40) ADAM17TGFBR1MMP2MMP3MMP7
SCHEMBL6946888 0.86 ADAM17 (0.48) ADAM17TGFBR1MMP1MMP2MMP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0993442-B1 HYDRAZINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2003-04-23 EP disclosed
US-6235787-B1 ANTIINFLAMMATORY AGENTS; RHEUMATIC DISEASES; BONE DISORDERS; SKIN DISORDERS; MULTIPLE SCLEROSIS HOFFMANN-LA ROCHE INC. 2001-05-22 US disclosed