SCHEMBL6944008

SCHEMBL6944008

Br[Mg]c1ccccc1.Clc1ccc([Mg]Br)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.48
CYP1A2 P05177 1/20 0.46
LMNA P02545 3/20 0.40
CYP2A6 P11509 1/20 0.40
CES2 O00748 1/20 0.38
CES1 P23141 1/20 0.38
ORAI1 Q96D31 1/20 0.38
ORAI2 Q96SN7 1/20 0.38
ORAI3 Q9BRQ5 1/20 0.38
TRPV6 Q9H1D0 1/20 0.38
L3MBTL1 Q9Y468 3/20 0.34
IDO1 P14902 2/20 0.34
TDO2 P48775 2/20 0.34
KDM4E B2RXH2 2/20 0.34
GAA P10253 1/20 0.34
SIGMAR1 Q99720 1/20 0.34
ADRA2A P08913 2/20 0.32
SLC6A2 P23975 2/20 0.32
SLC6A4 P31645 2/20 0.32
SLC6A3 Q01959 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23466995 0.89 LMNA (0.50) TSHRCYP1A2LMNACYP2A6CES2
SCHEMBL181194 0.89
Bromide SCHEMBL1272014 0.87 LMNA (0.47) TSHRCYP1A2LMNACYP2A6CES2
SCHEMBL5450 0.84
SCHEMBL11837452 0.82 CYP1A2 (0.48) TSHRCYP1A2LMNACYP2A6L3MBTL1
Water SCHEMBL5110307 0.81
Bromide SCHEMBL3131534 0.81
Water SCHEMBL6421934 0.81 ALDH1A1 (0.37) TSHRLMNATDP1MAPK1
Hydrochloric Acid SCHEMBL30169698 0.78 ALDH1A1 (0.35) TSHRTDP1
Ethyne SCHEMBL11077452 0.78 ALDH1A1 (0.35) TSHRTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1368299-A2 SUBSTITUTED C-CYCLOHEXYLMETHYLAMINE DERIVATIVES Grünenthal GmbH (DE) 2003-12-10 EP disclosed
WO-2002030870-A2 SUBSTITUTED C-CYCLOHEXYLMETHYLAMINE DERIVATIVES Grünenthal GmbH (DE) 2002-04-18 WO disclosed