SCHEMBL6944676

SCHEMBL6944676

Oc1ccc(OCCN2C3CCC2CC(Cc2ccccc2)C3)cc1

nearest known ligand 0.66

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TMEM97 Q5BJF2 2/20 0.52
SIGMAR1 Q99720 2/20 0.52
OPRM1 P35372 1/20 0.49
OPRD1 P41143 1/20 0.49
ESR1 P03372 2/20 0.47
ESR2 Q92731 2/20 0.47
LTA4H P09960 1/20 0.47
MAOB P27338 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6945442 0.88 ESR1 (0.44) TMEM97SIGMAR1ESR1ESR2LTA4H
SCHEMBL7402131 0.80 TMEM97 (0.82) TMEM97SIGMAR1LTA4HMAOB
SCHEMBL6947479 0.80 OPRM1 (0.59) OPRM1OPRD1
Hydrochloric Acid SCHEMBL7402650 0.79 TMEM97 (0.80) TMEM97SIGMAR1LTA4HMAOB
SCHEMBL6949983 0.78 OPRM1 (0.49) OPRM1OPRD1LTA4H
SCHEMBL6931066 0.75 TMEM97 (0.49) TMEM97SIGMAR1ESR1ESR2LTA4H
SCHEMBL7069836 0.75 TMEM97 (0.49) TMEM97SIGMAR1ESR1ESR2LTA4H
SCHEMBL6945483 0.72 OPRM1 (0.64) OPRM1OPRD1
SCHEMBL7246214 0.72 ESR1 (0.54) TMEM97SIGMAR1ESR1ESR2LTA4H
SCHEMBL12642496 0.72 LTA4H (0.49) OPRM1OPRD1ESR1ESR2LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1244450-A4 8-AZA-BICYCLO[3.2.1]OCTANE NMDA/NR2B ANTAGONISTS MERCK & CO INC (US) 2003-03-19 EP claimed
EP-1244450-A1 8-AZA-BICYCLO[3.2.1]OCTANE NMDA/NR2B ANTAGONISTS Merck & Co., Inc. (US) 2002-10-02 EP claimed
WO-2001032179-A1 8-AZA-BICYCLO[3.2.1]OCTANE NMDA/NR2B ANTAGONISTS MERCK & CO., INC. (US) 2001-05-10 WO claimed
EP-1244450-A4 8-AZA-BICYCLO[3.2.1]OCTANE NMDA/NR2B ANTAGONISTS MERCK & CO INC (US) 2003-03-19 EP disclosed
EP-1244450-A1 8-AZA-BICYCLO[3.2.1]OCTANE NMDA/NR2B ANTAGONISTS Merck & Co., Inc. (US) 2002-10-02 EP disclosed
US-6432976-B1 ANALGESICS; SIDE EFFECT REDUCTION MERCK & CO., INC. 2002-08-13 US disclosed
WO-2001032179-A1 8-AZA-BICYCLO[3.2.1]OCTANE NMDA/NR2B ANTAGONISTS MERCK & CO., INC. (US) 2001-05-10 WO disclosed