SCHEMBL6945353

SCHEMBL6945353

COC(Cc1ccc(CCCn2c(=O)c3ccccc3n(C)c2=O)cc1)C(N)=O

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TNF P01375 1/20 0.51
HDAC1 Q13547 5/20 0.46
HDAC6 Q9UBN7 4/20 0.41
HDAC8 Q9BY41 3/20 0.41
HDAC11 Q96DB2 2/20 0.41
ADORA3 P0DMS8 1/20 0.41
ADORA2B P29275 1/20 0.41
MAPT P10636 1/20 0.40
HDAC3 O15379 1/20 0.40
HDAC2 Q92769 1/20 0.40
ALDH1A1 P00352 1/20 0.39
TSHR P16473 1/20 0.39
TP53 P04637 2/20 0.39
ERCC1 P07992 1/20 0.39
FEN1 P39748 1/20 0.39
ERCC4 Q92889 1/20 0.39
MELK Q14680 1/20 0.39
PLA2G2A P14555 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6947459 0.91 TNF (0.52) TNFHDAC1HDAC6HDAC8HDAC11
SCHEMBL6952964 0.86 TNF (0.53) TNFHDAC1HDAC6HDAC8HDAC11
SCHEMBL7530431 0.75 PPARG (0.51)
SCHEMBL17241737 0.73 MAPT (0.63) TNFHDAC1HDAC6HDAC8HDAC11
SCHEMBL6952391 0.72 PPARG (0.46) TNFHDAC1HDAC6HDAC8HDAC11
SCHEMBL6947495 0.71 PPARA (0.46) ALDH1A1
SCHEMBL6510771 0.70 ERCC1 (0.60) TNFHDAC1ALDH1A1TSHRERCC1
SCHEMBL17241665 0.70 MAPT (0.56) TNFHDAC1HDAC6HDAC8HDAC11
SCHEMBL6956161 0.70 PPARG (0.46) TNFHDAC1HDAC6HDAC8HDAC11
SCHEMBL6953729 0.70 HTR1A (0.40) HDAC1MAPTALDH1A1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0903343-B1 Alpha-Substituted phenylpropionic acid derivative and medicine containing the same SSP CO LTD (JP) 2003-05-28 EP disclosed
EP-0903343-A1 Alpha-Substituted phenylpropionic acid derivative and medicine containing the same SSP Co., Ltd. (JP) 1999-03-24 EP disclosed