SCHEMBL6945565

SCHEMBL6945565

COc1cc[c]c(OCCc2cccc(Cl)c2Cl)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.39
CASR P41180 4/20 0.36
HTR1A P08908 3/20 0.35
ADRA2B P18089 1/20 0.35
ADRA2C P18825 1/20 0.35
SLC6A2 P23975 1/20 0.35
HRH2 P25021 1/20 0.35
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
HRH1 P35367 1/20 0.35
OPRM1 P35372 1/20 0.35
DRD3 P35462 1/20 0.35
OPRK1 P41145 1/20 0.35
HTR2B P41595 1/20 0.35
HTR5A P47898 1/20 0.35
HTR6 P50406 1/20 0.35
TMEM97 Q5BJF2 1/20 0.35
GPR65 Q8IYL9 1/20 0.35
SIGMAR1 Q99720 1/20 0.35
PNMT P11086 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5543377 0.75 TAAR1 (0.47) TAAR1PNMTIDO1MAPTL3MBTL1
SCHEMBL7953637 0.73 MAPK1 (0.40) MAPK1L3MBTL1SMN1; SMN2
SCHEMBL6554584 0.73 TUBB4A (0.39) MAPK1GAASMN1; SMN2
SCHEMBL7386281 0.71 ALDH1A1 (0.37) MAPK1SMN1; SMN2
SCHEMBL7387017 0.71 TAAR1 (0.39) TAAR1MAPK1ADRA1A
SCHEMBL29023056 0.71 CCR1 (0.34) MAPK1MAPT
SCHEMBL24822382 0.70 TAAR1 (0.57) TAAR1PNMTIDO1SMN1; SMN2HPGD
SCHEMBL1569511 0.69 ESR1 (0.39) MAPK1MAPTGAASMN1; SMN2ABCB1
SCHEMBL7389699 0.69 HTR1B (0.43) HTR2A
SCHEMBL7387972 0.69 MAPT (0.41) MAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1218739-A4 2-AMINOPYRIDINE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF LION BIOSCIENCE AG (DE) 2003-06-04 EP claimed
EP-1218739-A1 2-AMINOPYRIDINE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF TREGA BIOSCIENCES, INC. (US) 2002-07-03 EP claimed
WO-2001023887-A1 2-AMINOPYRIDINE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF LION BIOSCIENCE AG (DE) 2001-04-05 WO claimed